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Catalog | name | Description | price |
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R-R-1857 | Mepazine CAS No.60-89-9 | Mepazine (Pecazine)/CAS No.60-89-9 is a potent and selective MALT1 protease inhibitor with IC50s of 0.83 and 0.42 μM for GSTMALT1 full length and GSTMALT1 325-760, respectively. Mepazine affects viability of ABC-DLBCL cells by enhancing apoptosis. | price> |
R-CG-034 | PLGA-SS-PEG-Rhodamine B(RhB) | Poly(L-lactide-co-glycolide)-s-s-Polyethylene glycol-Rhodamine B(RhB),PLGA-SS-PEG-Rhodamine B(RhB) from ruixi.PLGA is connected with disulfide bond, then peg Rhodamine B(RhB)(PEG Rhodamine B(RhB) is coupled to form plga-s-s-peg-Rhodamine B(RhB).The product can be used to prepare micelles or vesicles and other new targeted products for drug encapsulation. | price> |
R-M-705 | Atosiban (free acid) trifluoroacetate salt | Atosiban (free acid) trifluoroacetate salt(CAS : 168102-69-0) is a Impurity and degradation product of atosiban. | price> |
R-R-1858 | Gemcitabine-13C,15N2 hydrochloride CAS No.2757566-59-7 | Gemcitabine-13C,15N2 (hydrochloride)/CAS No.2757566-59-7 is the 13C and 15N labeled Gemcitabine hydrochloride. Gemcitabine Hydrochloride (LY 188011 Hydrochloride) is a pyrimidine nucleoside analog antimetabolite and an antineoplastic agent. Gemcitabine Hydrochloride inhibits DNA synthesis and repair, resulting in autophagyand apoptosis. | price> |
R-CG-035 | PLGA-Hydrazone(hyd)-PEG-SH | Poly(L-lactide-co-glycolide)-s-s-Polyethylene glycol-SH,PLGA-SS-PEG-thiol from ruixi.Hydrazone bond has pH response effect. DSPE was linked to hydrazone bond and PEG thiol was coupled to form micelles with pH response. PH responsive polymer micelles can exist stably in normal tissue, but in the area of slightly acidic tumor tissue, the nucleus or shell of micelles undergo protonation or chemical reaction, which leads to the change of physical properties, the destruction of micelle structure, the rapid release of drugs from micelles to tumor tissue, and the better effect of killing cancer cells. | price> |
R-R-1859 | Mepazine hydrochloride CAS No.2975-36-2 | Mepazine hydrochloride (Pecazine hydrochloride)/CAS No.2975-36-2 is a potent and selective MALT1 protease inhibitor with IC50s of 0.83 and 0.42 μM for GSTMALT1 full length and GSTMALT1 325-760, respectively. Mepazine hydrochloride affects viability of ABC-DLBCL cells by enhancing apoptosis. | price> |
R-CG-036 | PLGA-Hydrazone(Hyd)-PEG-Azide(N3) | Poly(L-lactide-co-glycolide)-Hydrazone-Polyethylene glycol-Azide(N3),PLGA-Hyd-PEG-Azide(N3) from ruixi.Hydrazone bond has pH response effect. PLGA was linked to hydrazone bond and PEG Azide was coupled to form micelles with pH response. PH responsive polymer micelles can exist stably in normal tissue, but in the area of slightly acidic tumor tissue, the nucleus or shell of micelles undergo protonation or chemical reaction, which leads to the change of physical properties, the destruction of micelle structure, the rapid release of drugs from micelles to tumor tissue, and the better effect of killing cancer cells. | price> |
R-M-707 | BQ-788 sodium salt | BQ-788 sodium salt,CAS :156161-89-6 from ruixi.It is a synthetic peptide. | price> |
R-R-1860 | Bufarenogin CAS No.17008-65-0 | Bufarenogin/CAS No.17008-65-0 induces intrinsic apoptosis via Bax and ANT cooperation. | price> |
R-CG-037 | PLGA-Hydrazone(Hyd)-PEG-Alkyne | Poly(L-lactide-co-glycolide)-Hydrazone-Polyethylene glycol-Alkyne,PLGA-Hyd-PEG-Alkyne from ruixi.Hydrazone bond has pH response effect. PLGA was linked to hydrazone bond and PEG Alkyne was coupled to form micelles with pH response. PH responsive polymer micelles can exist stably in normal tissue, but in the area of slightly acidic tumor tissue, the nucleus or shell of micelles undergo protonation or chemical reaction, which leads to the change of physical properties, the destruction of micelle structure, the rapid release of drugs from micelles to tumor tissue, and the better effect of killing cancer cells. | price> |
R-M-708 | BQ-788 ammonium salt | BQ-788 ammonium salt,CAS : 173326-37-9 from ruixi.It is a synthetic peptide. | price> |
R-R-1861 | Taltobulin CAS No.228266-40-8 | Taltobulin (HTI-286)/CAS No.228266-40-8, a synthetic analogue of the tripeptide hemiasterlin, is a potent antimicrotubule agent that circumvents P-glycoprotein-mediated resistance in vitro and in vivo. Taltobulin inhibits the polymerization of purified tubulin, disrupts microtubule organization in cells, and induces mitotic arrest, as well as apoptosis. | price> |
R-CG-038 | PLGA-Hydrazone(Hyd)-PEG-oh | Poly(L-lactide-co-glycolide)-Hydrazone-Polyethylene glycol-hydroxyl,PLGA-Hyd-PEG-oh from ruixi.Hydrazone bond has pH response effect. PLGA was linked to hydrazone bond and PEG hydroxyl was coupled to form micelles with pH response. PH responsive polymer micelles can exist stably in normal tissue, but in the area of slightly acidic tumor tissue, the nucleus or shell of micelles undergo protonation or chemical reaction, which leads to the change of physical properties, the destruction of micelle structure, the rapid release of drugs from micelles to tumor tissue, and the better effect of killing cancer cells. | price> |
R-M-709 | BQ-788 | In vitro, BQ-788 potently and competitively inhibited ¹²⁵I-labeled ET-1 binding to ET-B receptors on human Girardi heart cells (IC₅₀= 1.2 nM). However, BQ-788 only poorly inhibited ET-1 binding to ET-A receptors on human neuroblastoma cell line SK-N-MC cells (IC₅₀= 1300 nM). Thus the ET-B receptor antagonist BQ788 may be considered as a powerful tool for investigating the role of ET in physiological and pathological processes. | price> |
R-R-1862 | Taltobulin hydrochloride | Taltobulin hydrochloride (HTI-286 hydrochloride), a synthetic analogue of the tripeptide hemiasterlin, is a potent antimicrotubule agent that circumvents P-glycoprotein-mediated resistance in vitro and in vivo. Taltobulin hydrochloride inhibits the polymerization of purified tubulin, disrupts microtubule organization in cells, and induces mitotic arrest, as well as apoptosis. | price> |
R-PL1052-X | PAMAM-PLGA-NH2 | Poly(amidoamine) -Poly(lactic-co-glycolic acid)-polyethylene glycol-Amine,PAMAM-PLGA-NH2 from ruixi.Poly(amidoamine) (PAMAM) dendrimers are a novel class of spherical, well-designed branching polymers with interior cavities and abundant terminal groups on the surface which can form stable complexes with drugs, plasmid DNA, oligonucleotides, and antibodies. PAMAM poly (lactide co glycolide) - amine, the dendrimer block copolymer of this product is a unique product of Ruixi biology. The product quality is high and the price is favorable. | price> |
R-M-710 | BQ-610 | BQ-610 is a very potent ET-A receptor antagonist which is about 30000 times more selective for ET-A receptors than for ET-B receptors. Furthermore, it has been found that BQ-610 strongly antagonizes ET-1 induced concentration in porcine coronary artery with a pA₂ value of 8.2. | price> |
R-R-1863 | Taltobulin trifluoroacetate CAS No.228266-41-9 | Taltobulin trifluoroacetate (HTI-286 trifluoroacetate)/CAS No.228266-41-9, a synthetic analogue of the tripeptide hemiasterlin, is a potent antimicrotubule agent that circumvents P-glycoprotein-mediated resistance in vitro and in vivo. Taltobulin trifluoroacetate inhibits the polymerization of purified tubulin, disrupts microtubule organization in cells, and induces mitotic arrest, as well as apoptosis. | price> |
R-R-1864 | Pladienolide B CAS No.445493-23-2 | Pladienolide B/CAS No.445493-23-2 is a potent cancer cell growth inhibitor that targets the SF3B1 subunit of the spliceosome. Pladienolide B exerts antitumor activities mediated through the inhibition of pre-mRNA splicing. Pladienolide B induces apoptosis. | price> |
R-CG-039 | PLGA-Hydrazone(Hyd)-PEG-CHO | Poly(L-lactide-co-glycolide)-Hydrazone-Polyethylene glycol-hydroxyl,PLGA-Hyd-PEG-CHO from ruixi.Hydrazone bond has pH response effect. PLGA was linked to hydrazone bond and PEG CHO was coupled to form micelles with pH response. PH responsive polymer micelles can exist stably in normal tissue, but in the area of slightly acidic tumor tissue, the nucleus or shell of micelles undergo protonation or chemical reaction, which leads to the change of physical properties, the destruction of micelle structure, the rapid release of drugs from micelles to tumor tissue, and the better effect of killing cancer cells. | price> |