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Catalog | name | Description | price |
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R-R-2862 | {Val1}-Exendin-3/4 | {Val1}-Exendin-3/4 is the first N-terminal 1-28 residues of Exendin-4 peptide. | price> |
R-C-1163 | OPC 21268 CAS:131631-89-5 | OPC21268 is a non-peptide AVP Receptor V(Vasopressin Receptor)antagonist that shows 1000-fold selectivity for V1 receptors over V2 receptors. | price> |
R-R-2863 | (1R,5S,6S)-Tert-butyl CAS No.:273206-92-1 | 6-amino-3-azabicyclo[3.1.0]hexane-3-carboxylate CAS No.:273206-92-1 The mode of action of (1R,5S,6S)-Tert-butyl 6-amino-3-azabicyclo[31It is known that the compound is synthesized via a palladium-catalyzed cyclopropanation of maleimides with n-tosylhydrazones . The interaction of this compound with its potential targets and the resulting changes are subjects of ongoing research. | price> |
R-C-1164 | GW9662 CAS: 22978-25-2 | GW9662 is a potent and selective PPARγ antagonist with an IC50 of 3.3 nM, showing 10 and 1000-fold selectivity over PPARα and PPARδ,respectively. | price> |
R-R-2864 | GLP-1 (1-36) amide (human, rat) (TFA) | GLP-1 (1-36) amide (human, rat) (Glucagon-like Peptide 1 (1-36) amide (human, rat) ) TFA is a molecular variant of glucagon-like peptide 1 (GLP-1)-(7-36) amide. GLP-1 (1-36) amide (human, rat) TFA can stimulate [14C]aminopyrine accumulation on enzymatically dispersed enriched rat parietal cells. | price> |
R-C-1165 | Coelenterazine H CAS:50909-86-9 | Coelenterazine h is a derivative of Coelenterazine.Coelenterazine h is more sensitive to Ca2+than is the native complex,thus providing a valuable tool for measuring small changes in Ca2+concentrations. | price> |
R-R-2865 | SAR441255 TFA | SAR441255 TFA is a potent unimolecular peptide GLP-1/GIP/GCG receptor triagonist. SAR441255 TFA displays high potency with balanced activation of all three target receptors.?SAR441255 TFA shows positive acute glucoregulatory effectss in diabetic obese monkeys. | price> |
R-C-1166 | AI-10-49 CAS:1256094-72-0 | AI-10-49 is a protein-protein interaction inhibitor that selectively binds to CBFβ-SMMHC and disrupts its binding to RUNX1 with a FRET IC50 of 0.26 uM. | price> |
R-R-2866 | V-0219 CAS No.878453-71-5 | V-0219 (Compound 9)/CAS No.878453-71-5 is an orally active, positive allosteric modulator (PAM) of the glucagon-like peptide-1 receptor (GLP-1R). V-0219 can be used for obesity-associated diabetes research. | price> |
R-C-1167 | Tideglusib (NP031112, NP-12) CAS:865854-05-3 | Tideglusib(NP031112)is an irreversible GSK-3 inhibitor with IC50s of 5 nM and 60 nM for GSK-3βWT(1 h preincubation)and GSK-3βC199A(1 h preincubation), respectively. | price> |
R-R-2867 | V-0219 hydrochloride CAS No.2922283-73-4 | V-0219 hydrochloride (Compound 9)/CAS No.2922283-73-4 is an orally active, positive allosteric modulator (PAM) of the glucagon-like peptide-1 receptor (GLP-1R). V-0219 hydrochloride can be used for obesity-associated diabetes research. | price> |
R-C-1168 | Elesclomol (STA-4783) CAS: 488832-69-5 | Elesclomol(STA-4783)is an oxidative stress inducer that induces cancer cell apoptosis.Elesclomol is a reactive oxygen species(ROS)inducer.Elesclomol shows antitumor activity against a broad range of cancer cell types.Elesclomol is also a highly lipophilic Cu2+-binding molecule.Elesclomol can be used for Menkes and associated disorders of hereditary copper deficiency research. | price> |
R-R-2868 | Apraglutide TFA | Apraglutide TFA (FE 203799 TFA), a synthetic 33-amino-acid peptide and a long-acting GLP-2 analogue, enhances adaptation and linear intestinal growth in a neonatal piglet model of short bowel syndrome with total resection of the ileum. | price> |
R-C-1169 | GW 627368 CAS: 439288-66-1 | GW627368(GW627368X)is a novel,potent and selective competitive antagonist of prostanoid EP4 receptor with additional human TP receptor affinity, with pKi values of 7.0 and 6.8 for human prostanoid EP4 and TP receptors respectively. | price> |
R-R-2869 | (S)-V-0219 hydrochloride | (S)-V-0219 hydrochloride is an enantiomer of V-0219 (HY-143312). V-0219 is an orally active and positive allosteric modulator (PAM) of the GLP Receptor-1 (GLP-1R). (S)-V-0219 hydrochloride activates calcium fluxes in HEK cells stably expressing hGLP-1R. (S)-V-0219 hydrochloride is orally active and ameliorates high glucose levels in mice and inhibits feeding behavior in fasted mice. | price> |
R-C-1170 | cevipabulin CAS:849550-05-6 | Cevipabulin(TTI-237),an antimicrotubule agent,is a small synthetic molecule of triazolopyrimidine derivative with potential antitumor activity.With a novel mechanism of action distinct from the action of other vinca alkaloid compounds, TTI-237 specifically binds to tubulin at the vinca site,and promotes the polymerization of tubulin into microtubules. | price> |
R-R-2870 | GLP-1 receptor agonist 11 CAS No.2784590-83-4 | GLP-1 receptor agonist 11 (compound 3)/CAS No.2784590-83-4 is an agonist of GLP Receptor. GLP-1 receptor agonist 11 can be used in the study of diseases such as diabetes and non-alc. fatty liver disease. | price> |
R-C-1171 | LY2874455 CAS:1254473-64-7 | LY2874455 is a pan-FGFR inhibitor with IC50 of 2.8 nM,2.6 nM,6.4 nM,and 6 nM for FGFR1,FGFR2,FGFR3,and FGFR4,respectively,and also inhibits VEGFR2 activity with IC50 of 7 nM. | price> |
R-R-2871 | (R)-V-0219 hydrochloride | (R)-V-0219 hydrochloride is an enantiomer of V-0219 (HY-143312). V-0219 is an orally active and positive allosteric modulator (PAM) of the GLP Receptor-1 (GLP-1R). (R)-V-0219 hydrochloride activates calcium fluxes in HEK cells stably expressing hGLP-1R. | price> |
R-C-1172 | BLU-9931 CAS:1538604-68-0 | BLU9931 is a potent,highly selective,and irreversible fibroblast growth factor receptor 4(FGFR4)inhibitor with an IC50 of 3 nM and a Kd of 6 nM.BLU9931 has significant antitumor activity. | price> |