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Catalog	name	Description	price
R-C-2073	Oxaliplatin CAS：61825-94-3	Oxaliplatin is an organoplatinum complex in which the platinum atom is complexed with 1,2-diaminocyclohexane(DACH)and with an oxalate ligand as a leaving group.A leaving group is an atom or a group of atoms that is displaced as a stable species taking with it the bonding electrons.The DACH side chain appears to inhibit alkylating-agent resistance.	price>
R-R-3773	Zinc(II) Tetraphenylporphyrin CAS :14074-80-7	Zinc(II) Tetraphenylporphyrin/CAS :14074-80-7 is a natural organic compound that can be found in the human body. It has been shown to have anti-angiogenic properties and can be used for the treatment of choroidal neovascularization (CNV). Tetraphenylporphyrin is a redox active molecule that has a high redox potential, which makes it an ideal candidate for use in photoactive systems. Tetraphenylporphyrin has been shown to inhibit the proliferation of tumor cells by interfering with lipid synthesis and transferring electrons from one molecule to another. The chemical structure of tetraphenylporphyrin makes it possible for light exposure to induce a frequency shift, which leads to light emission at 590 nm. This emission is due to the hydroxyl group present on tetraphenylporphyrin, which acts as an electron donor. We can mass produce (kg level), process scaling up, pilot supply, raw material supply, and intermediate production. Our production technology is mature and more cost-effective. Feel free to inquire at any time.	price>
R-C-2074	CCT245737 CAS：1489389-18-5	CCT245737 is a potent, selective and orally active checkpoint kinase 1(CHK1) inhibitor.CCT245737 showed CHK1 IC50=1.3nM,CHK2 IC50=2440nM,G2 check point abrogation IC50=30nM.Mouse F(oral)=100%.CCT245737 demonstrated a favorable physicochemical,PK,and PD-efficacy profile.The serine-threonine kinase CHK1 is a critical component of the cellular response to DNA damage,especially the repair of DNA breaks arising during replication or caused by DNA damaging chemotherapies and ionizing radiation.	price>
R-R-3774	Terazosin hydrochloride CAS No.63074-08-8	Terazosin hydrochloride/CAS No.63074-08-8 is a quinazoline derivative and a competitive and orally active α1-adrenoceptor antagonist. Terazosin hydrochloride works by relaxing blood vessels and the opening of the bladder. Terazosin hydrochloride has the potential for benign prostatic hyperplasia (BPH) and high blood pressure treatment.	price>
R-C-2075	SJB2-043 CAS：63388-44-3	SJB2-043 is one of analogs/derivatives of C527,which is a novel and potent USP1 (ubiquitin-specific protease 1)inhibitor.	price>
R-R-3775	Levobunolol hydrochloride CAS No.27912-14-7	Levobunolol (l-Bunolol) hydrochloride/CAS No.27912-14-7 is a potent and nonselective β-adrenergic receptor antagonist. Levobunolol hydrochloride is an ocular hypotensive agent and lowers mean intraocular pressure (IOP). Levobunolol hydrochloride can be used for glaucoma and superior oblique myokymia (SOM) research.	price>
R-C-2076	SU14813 CAS： 627908-92-3	SU14813 is a multi-targeted receptor tyrosine kinases inhibitor with IC50s of 50,2,4,15 nM for VEGFR2,VEGFR1,PDGFRβ and KIT.	price>
R-R-3776	Isoferulic acid CAS No.537-73-5	Isoferulic acid (3-Hydroxy-4-methoxycinnamic acid)/CAS No.537-73-5 is a cinnamic acid derivative that has antidiabetic activity. Isoferulic acid binds to and activates α1-adrenergic receptors (IC50=1.4 µM) to enhance secretion of β-endorphin (EC50=52.2 nM) and increase glucose use. Isoferulic acid also has anti-influenza virus activities.	price>
R-R-3777	Medetomidine CAS No.86347-14-0	Medetomidine/CAS No.86347-14-0 is an orally active α2-adrenoceptor agonist (Ki: 1.08 nM). Medetomidine has sedative and analgesic effects. Medetomidine can cause peripheral vasoconstriction through the activation of α2 adrenoceptors on blood vessels.	price>
R-C-2078	Fmoc-Ser(Ac3GalNAcα)-OH CAS：120173-57-1	Fmoc-Ser(O-α-D-GalNAc(OAc)3)-OH is a drug for cancer.	price>
R-R-3778	Bevantolol hydrochloride CAS No.42864-78-8	Bevantolol hydrochloride/CAS No.42864-78-8 is a selective β1 and α1-adrenergic receptor antagonist with pKi values of 7.83, 6.9 in rat cerebral cortex, respectively. Bevantolol hydrochloride is a potent Ca2+ antagonist.	price>
R-C-2079	E-7046 CAS：1369489-71-3	E7046 is an orally bioavailable and specific EP4 antagonist,with IC50 of 13.5nM and Ki of 23.14nM,exhibiting anti-tumor activities.	price>
R-R-3779	Bambuterol hydrochloride CAS No.81732-46-9	Bambuterol hydrochloride/CAS No.81732-46-9 ((±)-Bambuterol hydrochloride; KWD-2183 hydrochloride) is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; it also is a proagent of terbutaline.	price>
R-C-2080	Bemcentinib (R428) CAS：1037624-75-1	Bemcentinib(R428,BGB324)is an inhibitor of Axl with IC50 of 14 nM,>100-fold selective for Axl versus Abl.Selectivty for Axl is also greater than Mer and Tyro3(50-to-100- fold more selective)and InsR,EGFR,HER2,and PDGFRβ(100- fold more selective).	price>
R-R-3780	Dabuzalgron CAS No.219311-44-1	Dabuzalgron (Ro 115-1240)/CAS No.219311-44-1 is an orally active and selective α-1A adrenergic receptor agonist for the treatment of urinary incontinence. Dabuzalgron protects against Doxorubicin-induced cardiotoxicity by preserving mitochondrial function.	price>
R-C-2081	CPI-444 CAS：1202402-40-1	Ciforadenant(CPI-444,V81444)is a potent and selective Adenosine A2A receptor antagonist.It binds to A2A receptors with a Ki of 3.54 nmol/L and demonstrates a greater than 50-fold selectivity for the A2A receptor over other adenosine receptor subtypes.	price>
R-R-3781	Esmolol hydrochloride CAS No.81161-17-3	Esmolol hydrochloride/CAS No.81161-17-3 is a beta adrenergic receptor blocker.	price>
R-C-2082	ars-1620 CAS：1698055-85-4	ARS-1620 is a potent,orally bioavailable covalent inhibitor of KRAS-G12C and could achieve rapid and sustained in vivo target occupancy to induce tumor regression.	price>
R-R-3782	Glaucine CAS No.475-81-0	Glaucine (O,O-Dimethylisoboldine)/CAS No.475-81-0 is an alkaloid isolated from Glaucium flavum with antitussive, bronchodilation and anti-inflammatory properties. Glaucine is a selective and orally active phosphodiesterase 4 (PDE4) inhibitor with Kis of 3.4 µM in human bronchus and polymorphonuclear leukocytes. Glaucine is also a non-selective α-adrenoceptor antagonist, a Ca2+ entry blocker, and a weak dopamine D1 and D2 receptor antagonist. Glaucine has antioxidative and antiviral activities.	price>
R-C-2083	USP25 and 28 inhibitor AZ-1 CAS：2165322-94-9	USP25/28 inhibitor AZ1(AZ1)is an orally active,selective,noncompetitive, dual ubiquitin specific protease(USP)25/28 inhibitor with IC50s of 0.7μM and 0.6 μM,respectively.USP25/28 inhibitor AZ1 attenuates colitis and tumorigenesis in the mice model.	price>

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