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Catalog	name	Description	price
R-R-3957	ST91 CAS No.4749-61-5	ST91/CAS No.4749-61-5 is a α2-adrenoceptor (α2AR) agonist. ST91 activates both α2AAR and non-α2AAR subtypes to produce spinal antinociception.	price>
R-R-3958	Octopamine-d4 hydrochloride CAS No.1219803-62-9	Octopamine-d4 (hydrochloride)/CAS No.1219803-62-9 is the deuterium labeled Octopamine hydrochloride. Octopamine ((±)-p-Octopamine) hydrochloride, a biogenic monoamine structurally related to noradrenaline, acts as a neurohormone, a neuromodulator and a neurotransmitter in invertebrates. Octopamine hydrochloride can stimulate alpha2-adrenoceptors (ARs) in Chinese hamster ovary cells transfected with human alpha2-ARs. Octopamine hydrochloride increased glycogenolysis, glycolysis, oxygen uptake, gluconeogenesis and the portal perfusion pressure.	price>
R-R-3959	Amitriptyline hydrochloride (Standard) CAS No.549-18-8	Amitriptyline (hydrochloride) (Standard)/CAS No.549-18-8 is the analytical standard of Amitriptyline (hydrochloride). This product is intended for research and analytical applications. Amitriptyline hydrochloride is an inhibitor of serotonin reuptake transporter (SERT) and noradrenaline reuptake transporter (NET), with Kis of 3.45 nM and 13.3 nM for human SERT and NET, respectively. Amitriptyline hydrochloride also weakly binds to dopamine reuptake transporter (DAT) with a Ki of 2.58 μM. Amitriptyline hydrochloride also inhibits adrenergic, muscarinic, histamine and 5-HT receptors. Amitriptyline hydrochloride is a TrkA and TrkB receptors agonist with potent neurotrophic activity. Amitriptyline hydrochloride has antidepressant activity.	price>
R-R-3960	Butyryltimolol CAS No.106351-79-5	Butyryltimolol/CAS No.106351-79-5, an effective precursor of Timolol, improves the corneal penetration of Timolol. Butyryltimolol is a β-adrenergic blocker.	price>
R-R-3961	Prazosin-d8 hydrochloride CAS No.1189508-34-6	Prazosin-d8 hydrochloride/CAS No.1189508-34-6 is the deuterium labeled Prazosin hydrochloride. Prazosin hydrochloride is an alpha-adrenergic blocker.	price>
R-R-3962	Piribedil-d8 CAS No.1398044-45-5	Piribedil-d8/CAS No.1398044-45-5 is the deuterium labeled Piribedil, which is an antiparkinsonian agent.	price>
R-R-3963	Carazolol-d7 CAS No.1173021-02-7	Carazolol-d7/CAS No.1173021-02-7 is the deuterium labeled Carazolol.	price>
R-R-3964	Mirtazapine-d4 CAS No.1215898-55-7	Mirtazapine-d4/CAS No.1215898-55-7 is deuterium labeled Mirtazapine. Mirtazapine (Org3770) is a potent and orally active noradrenergic and specific serotonergic antidepressant (NaSSA) agent. Mirtazapine is also a 5-HT2, 5-HT3, histamine H1 receptor and α2-adrenoceptor antagonist with pKi values of 8.05, 8.1, 9.3 and 6.95, respectively.	price>
R-C-2265	Ribociclib hydrochloride CAS：1211443-80-9	Ribociclib hydrochloride(LEE011 hydrochloride)is a highly specific CDK4/6 inhibitor with IC50 values of 10nM and 39nM,respectively,and is over 1,000-fold less potent against the cyclin B/CDK1 complex.	price>
R-R-3965	Clorprenaline-d6 CAS No.1648796-40-0	Clorprenaline-d6/CAS No.1648796-40-0 is the deuterium labeled Clorprenaline.	price>
R-C-2266	Pemetrexed (LY-231514) disodium CAS:150399-23-8	Pemetrexed(LY-231514)disodium is a novel antifolate and antimetabolite for TS,DHFR and GARFT with Ki of 1.3nM,7.2nM and 65nM in cell-free assays, respectively.Pemetrexed induces autophagy and apoptosis.	price>
R-R-3966	Clencyclohexerol CAS No.157877-79-7	Clencyclohexerol/CAS No.157877-79-7 is a β-agonist. Clencyclohexerol can be used as a growth promoter in animals.	price>
R-C-2267	SCR130 CAS: 2377858-38-1	SCR130 is a novel DNA repair inhibitor with IC50s of 14μM in Reh cells and 2μM in Nalm6 cells.SCR130 specifically inhibits DNA Ligase IV mediated joining with minimal or no effect on Ligase III and Ligase I mediated joining.	price>
R-R-3967	Phenylethanolamine A-d3 CAS No.2507994-61-6	Phenylethanolamine A-d3/CAS No.2507994-61-6 is a deuterium labeled Phenylethanolamine A. Phenylethanolamine A acts as a β-adrenergic agonist. Phenylethanolamine A is a byproduct during the Ractopamine synthesis process.	price>
R-C-2268	PFM01 CAS:1558598-41-6	PFM01,N-alkylated Mirin derivative,is a MRE11 endonuclease inhibitor.PFM01 can regulate double-strand break repair(DSBR)by nonhomologous end-joining (NHEJ)versus homologous recombination(HR).	price>
R-R-3968	Carvedilol (Standard) CAS No.72956-09-3	Carvedilol (Standard)/CAS No.72956-09-3 is the analytical standard of Carvedilol. This product is intended for research and analytical applications. Carvedilol (BM 14190) is a non-selective β/α-1 blocker. Carvedilol inhibits lipid peroxidation in a dose-dependent manner with an IC50 of 5 μM. Carvedilol is a multiple action antihypertensive agent with potential use in angina and congestive heart failure. Carvedilol is an autophagy inducer that inhibits the NLRP3 inflammasome.	price>
R-C-2269	Metarrestin (ML246) CAS:1443414-10-5	Metarrestin(ML246)is an orally active and specific perinucleolar compartment (PNC)inhibitor that disrupts the nucleolar structure and inhibits RNA polymerase(Pol)I transcription.Metarrestin blocks metastatic development and extends survival in mouse cancer models.	price>
R-R-3969	Betaxolol-d5 CAS No.1189957-99-0	Betaxolol-d5/CAS No.1189957-99-0 is the deuterium labeled Betaxolol. Betaxolol is a selective beta1 adrenergic receptor blocker that can be used for the research of hypertension and glaucoma.	price>
R-C-2270	Menthone CAS:10458-14-7	Menthone is one of the main volatile components of the essential oil of peppermint (Mentha piperita L.).Menthone is used as antioxidant agent and has a good compensatory effect with significant reduction in DNA damages in sperm cells.	price>
R-R-3970	HEAT hydrochloride CAS No.30007-39-7	HEAT (BE2254) hydrochloride/CAS No.30007-39-7 is a selective alpha 1 adrenergic receptor antagonist. HEAT hydrochloride, a phenethylamine derivative, shows pKis of 9, 9.1, and 8.57 for alpha 1a, alpha 1b and alpha 1c, respectively.	price>

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