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Catalog | name | Description | price |
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R-R-4836 | 7-Methylguanosine CAS No.20244-86-4 | 7-Methylguanosine/CAS No.20244-86-4 is a novel cNIIIB nucleotidase inhibitor with IC50 value of 87.8 ± 7.5 µM. | price> |
R-C-3167 | NCRW0005-F05 CAS:342779-66-2 | NCRW0005-F05, first antagonist selective for GPR139 (IC50 value 0.21 uM); a useful tool to study GPR139 pharmacology, especially in combination with the GPR139 agonist JNJ 63533054.Our products are only suitable for scientific research experiments, not for clinical experiments and human body. | price> |
R-R-4837 | Sangivamycin CAS No.18417-89-5 | Sangivamycin (NSC 65346)/CAS No.18417-89-5, a nucleoside analog, is a potent inhibitor of protein kinase C (PKC) with an Ki of 10 μM. Sangivamycin has potent antiproliferative activity against a variety of human cancers. | price> |
R-C-3168 | BMS-564929 CAS:627530-84-1 | BMS-564929 is a novel, highly potent, orally active, nonsteroidal tissue selective androgen receptor (AR) modulator, and this compound has been advanced to clinical trials for the treatment of age-related functional decline. Our products are only suitable for scientific research experiments, not for clinical experiments and human body. | price> |
R-R-4838 | 3-Methylcytidine CAS No.2140-64-9 | 3-Methylcytidine/CAS No.2140-64-9, a urinary nucleoside, can be used as a biomarker of four different types of cancer: lung cancer, gastric cancer, colon cancer, and breast cancer. | price> |
R-C-3169 | AZD3514 CAS:1240299-33-5 | AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2M and has ability of reducing AR protein expression.Our products are only suitable for scientific research experiments, not for clinical experiments and human body. | price> |
R-R-4839 | 6-Thioinosine CAS No.574-25-4 | 6-Thioinosine (6TI)/CAS No.574-25-4 is a purine antimetabolite, acts as an anti-adipogenesis agent, downregulates mRNA levels of PPAR γ and C/EBPα, as well as PPAR γ target protein such as LPL, CD36, aP2, and LXRα. | price> |
R-C-3170 | GSK-2881078 CAS :1539314-06-1 | GSK 2881078 is a nonsteroidal selective modulator of androgen receptor that is potentially used for the treatment of cachexia.Our products are only suitable for scientific research experiments, not for clinical experiments and human body. | price> |
R-R-4840 | N2-Methylguanosine CAS No.2140-77-4 | N2-methylguanosine/CAS No.2140-77-4 is a modified nucleoside that occurs at several specific locations in many tRNAs. | price> |
R-C-3171 | MK-0773 CAS: 606101-58-0 | MK-0773,one of selective androgen receptor modulators(SARMs),is a 4-aza-steroid that exhibited tissue selectivity in humans (IC50=6.6nM).Our products are only suitable for scientific research experiments, not for clinical experiments and human body. | price> |
R-R-4841 | 3-Deazauridine CAS No.23205-42-7 | 3-Deazauridine (NSC 126849)/CAS No.23205-42-7 is a uridine analogue. 3-Deazauridine competitively inhibits cytidine triphosphate synthase to inhibit the biosynthesis of cytidine-5-triphosphate. 3-Deazauridine acts synergistically with several antineoplastic agents, acting as a biological response modifier. | price> |
R-C-3172 | EPI-001 CAS:227947-06-0 | EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ∼6μM and a selective PPAR-gamma modulator.Our products are only suitable for scientific research experiments, not for clinical experiments and human body. | price> |
R-R-4842 | Peldesine dihydrochloride CAS No.2772702-10-8 | Peldesine (BCX 34) dihydrochloride/CAS No.2772702-10-8 is a potent, competitive, reversible and orally active purine nucleoside phosphorylase (PNP) inhibitor with IC50s of 36 nM, 5 nM, and 32 nM for human, rat, and mouse red blood cell (RBC) PNP, respectively. Peldesine dihydrochloride is also a T-cell proliferation inhibitor with an IC50 of 800 nM. Peldesine dihydrochloride has the potential for cutaneous T-cell lymphoma, psoriasis and HIV infection research. | price> |
R-C-3173 | Tanaproget CAS:304853-42-7 | Tanaproget is a novel nonsteroidal progesterone receptor agonist which can bind to the PR from various species with a higher relative affinity than reference steroidal progestins.Our products are only suitable for scientific research experiments, not for clinical experiments and human body. | price> |
R-R-4843 | 2-Deoxy-2-fluoro-5-iodouridine CAS No.55612-21-0 | 2-Deoxy-2-fluoro-5-iodouridine/CAS No.55612-21-0 is a purine nucleoside analog. Purine nucleoside analogs have broad antitumor activity targeting indolent lymphoid malignancies. Anticancer mechanisms in this process rely on inhibition of DNA synthesis, induction of apoptosis, etc. | price> |
R-C-3174 | ACT-129968 (Setipiprant) CAS:866460-33-5 | Setipiprant is an orally available,selective CRTH2 antagonist. Our products are only suitable for scientific research experiments, not for clinical experiments and human body. | price> |
R-R-4844 | HOF-5 | HOF-5/hydrogen bonded organic framework material-5 is a Hydrogen bonded organic Framewok (HOF for short) material. The specific synthesis method and chemical structure of HOF-5 may vary among researchers and laboratories. However, generally speaking, HOFs are formed through hydrogen bonding interactions between organic molecules, and these hydrogen bonds play a key role in the framework structure, giving it a high degree of order and stability. Due to the special structure and properties of HOFs, they have potential application value in the fields of gas adsorption and separation, catalysis, chemical sensing, and drug delivery. In addition, HOF; can also be functionalized through post-modification and other methods to further expand its application fields. | price> |
R-C-3175 | Etonogestrel CAS:54048-10-1 | Etonogestrel (Implanon, Nexplanon,3-Oxodesogestrel,3-keto-Desogestrel) is a synthetic form of the naturally occurring female sex hormone progesterone.It binds to the cytoplasmic progesterone receptors in the reproductive system and subsequently activates progesterone receptor mediated gene expression.Our products are only suitable for scientific research experiments, not for clinical experiments and human body. | price> |
R-R-4845 | MOF-818 | MOF-818/Metal-organic framework-818 is a metal-organic framework (MOf) material with a trinuclear copper center. It was first reported by LI et al. and found that it can simulate the activity of natural phenol oxidase with copper active sites. MOF-818 can efficiently catalyze the conversion of catechol into o-quinone and does not exhibit obvious peroxidase activity, which indicates the specificity of its catalytic process. Regarding the specific application of MOF-818, there has not yet been extensive research and reporting. However, due to its ability to simulate the activity of natural enzymes, it may have certain application potential in biochemistry, medicine, environmental science and other fields. For example, it can be used as a biocatalyst for drug synthesis, biosensors, environmental management, etc. In addition, the structure and properties of MOF-818 can be optimized through further modification and regulation to improve its catalytic activity and stability. This may require more research work and experimental validation. | price> |
R-R-4846 | COM-ETTA-BPDA | COM-ETTA-BPDA is a metal organic framework (Metahorganic Framewok, MOF for short) material, also known as Uio-66NH2. It is a three-dimensional porous structure constructed from zr6+ ions, terephthalic acid (BPDA) and ethylenediaminetetraacetic acid (ETTA) through coordination.COM-ETTA-BPDA combines the advantages of UIO-66-NH2 such as high stability, large specific surface area and good chemical stability, and introduces ethylenediaminetetraacetic acid (ETTA) as a connecting agent to increase the functional groups and activity of the material. site. This makes COM-ETTA-BPDA have broad application prospects in the fields of gas adsorption and separation, catalysis, chemical sensing, drug delivery, and bioimaging. For example, COM-ETTA-BPDA can be used as an efficient gas adsorbent to separate and purify carbon dioxide, methane and other gases in the air. In addition, its porous structure and abundant functional groups make it an excellent catalyst support that can be used to catalyze various organic reactions. At the same time, COM-ETTA-BPDA can also be used as a fluorescent probe in fields such as biological imaging and chemical sensing. | price> |