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Catalog	name	Description	price
R-R-2549	PBRM1-BD2-IN-8 CAS No.2819989-75-6	PBRM1-BD2-IN-8 (compound 34)/CAS No.2819989-75-6 is a potent PBRM1 Bromodomain inhibitor (PBRM1-BD2 Kd=4.4 μM, PBRM1-BD2 IC50=0.16 μM; PBRM1-BD5 Kd=25 μM). PBRM1-BD2-IN-8 shows anti-cancer activity.	price>
R-C-850	DPA-PEG-DPA	Dopamine is the most abundant catecholamine neurotransmitter in the brain.It is a neurotransmitter,a chemical that helps cells deliver pulses.This kind of secretion in the brain is related to people lust and feeling,It conveys the information of excitement and happiness.Polyethylene glycol(PEG)is a polymer of ethylene oxide hydrolysatewhich is non-toxic and non irritating.It is widely used in various pharmaceutical preparations.	price>
R-R-2550	GSK4028 CAS No.2079886-19-2	GSK4028/CAS No.2079886-19-2 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4.9 in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay.	price>
R-C-851	MC (C5)-Val-Cit	MC(C5)-Val CIT is a kind of cleavable ADC linker,which can be used to synthesize antibody coupled drugs(ADC).	price>
R-R-2551	BRM/BRG1 ATP Inhibitor-2 CAS No.2368900-77-8	BRM/BRG1 ATP Inhibitor-2/CAS No.2368900-77-8 is a BRG1/BRM ATPase inhibitor for the research of BAF-related disorders.	price>
R-C-852	Peptide-PEG2K-upconversion materia（NaGdF4：Yb,Er@NaGdF4）	The core-shell NaGdF4:Yb,Er@NaGdF4,nd upconversion nanoparticles(ucnps)were successfully prepared by polypeptide peg2k upconversion material coprecipitation method.The water solubility of ucnps was improved by ligand exchange reaction between nitrous groups of tetrafluoroborate.	price>
R-R-2552	PROTAC BRD4 Degrader-8	PROTAC BRD4 Degrader-8 is a PROTAC connected by ligands for von Hippel-Lindau and BRD4, with IC50s of 1.1 nM and 1.4 nM for BRD4 BD1 and BD2, respectively. PROTAC BRD4 Degrader-8 is capable of potently degrading the BRD4 protein in PC3 prostate cancer cells.	price>
R-C-853	FeCo-TCPP	TCPP(tris(1-chloro-2-propyl)phosphate)is a flame retardant commonly used in polyurethane foam in consumer products and in home insulation,and in electronics.It is used as an additive to polyurethane foam and is not chemically bound,and it escapes from products into the indoor environment.	price>
R-R-2553	LT052 CAS No.2543545-44-2	LT052/CAS No.2543545-44-2 is a highly selective BET BD1 inhibitor with an IC50 of 87.7 nM. LT052 exhibits nanomolar BRD4 BD1 potency and 138-fold selectivity over BRD4 BD2 (IC50=12.130 μM). LT052 has anti-inflammatory activity and can be used for acute gout arthritis research.	price>
R-C-854	PGA100-NH2	Polyglutamic acid(γ-PGA),also known as natto gum and polyglutamic acid,is a kind of water-solublebiodegradable,non-toxic biopolymer produced by microbial fermentation.	price>
R-R-2554	BETd-246 CAS No.2140289-17-2	BETd-246/CAS No.2140289-17-2 is a second-generation and PROTAC-based BET bromodomain (BRD) inhibitor connected by ligands for Cereblon and BET, exhibiting superior selectivity, potency and antitumor activity.	price>
R-C-855	Fruquintinib	Fruquintinib is an orally available,small molecule inhibitor of vascular endothelial growth factor receptors(VEGFRs),with potential anti-angiogenic and antineoplastic activities.	price>
R-R-2555	PROTAC BET degrader-3	PROTAC BET Degrader-3 is a PROTAC connected by ligands for von Hippel-Lindau and BET.	price>
R-C-856	Succinate vitamin E-PEI1.8k-mannose	Vitamin E succinate(RRR-α-tocopheryl succinate,VES)is an esterified derivative of vitamin E.Vitamin E is one of the most effective anti-tumor compounds,but it has no obvious anti-tumor effect.	price>
R-R-2556	LP99 CAS No.1808951-93-0	LP99/CAS No.1808951-93-0, an epigenetic probe, is a potent and selective inhibitor of the BRD7 and BRD9 bromodomains with a Kd of 99 nM against BRD9. LP99 disrupts the binding of BRD7 and BRD9 to chromatin in cells.	price>
R-C-857	5-hydroxydopamine-cisplatin-5-hydroxydopamine	Cisplatin(CDDP)is a platinum containing anticancer drug,namely CIS dichlorodiamine combined with platinum(II).Its brownish yellow powder is a cell cycle nonspecific drug.It has therapeutic effect on sarcoma,malignant epithelial tumor,lymphoma and germ cell tumor.	price>
R-R-2557	RVX-297 CAS No.1044871-04-6	RVX-297/CAS No.1044871-04-6 is a potent, orally active BET bromodomain inhibitor with selectivity for BD2. RVX-297 shows IC50s of 0.08, 0.05, and 0.02 μM for BRD2(BD2), BRD3(BD2), and BRD4(BD2), respectively. RVX-297 suppresses inflammatory gene expression in multiple immune cell types. RVX-297 is effective in acute inflammation and autoimmunity models.	price>
R-C-858	SUPER FLUOR 555-NHS	Cyanine dyes and their derivatives are often used in biological molecular labeling,fluorescence imaging and other fluorescent biological analysis.They are widely used to label peptides,proteins and nucleic acids.Cy7 is a near infrared cyanine dye.	price>
R-R-2558	Bleximenib oxalate CAS No.2866179-95-3	Bleximenib oxalate/Menin-MLL inhibitor 24 (compound A) oxalate/CAS No.2866179-95-3 is a menin-mixed-lineage leukemia 1 (menin-MLL) inhibitor, and can be used for the research of cancer.	price>
R-C-859	Alexa Fluor 488	Alexa fluor 488 is a kind of bright green fluorescent dye,and its excitation is very suitable for 488 nm laser line.In order to generate stable signals in imaging and flow cytometry,Alexa fluor 488 dye is not sensitive to pH in a wide range of moles.The probe with high fluorescence quantum yield and high photostability can detect low abundance biological structures with high sensitivity.Alexa-fluor488 dye molecules can attach to proteins at high molar ratio without significant self quenching,thus achieving brighter binding and more sensitive detection.	price>

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