Home > Keywords >
Catalog | name | Description | price |
---|---|---|---|
R-C-1130 | TAK063 CAS:1238697-26-1 | TAK-063,also known as Balipodect.,is a highly potent,selective,and orally active phosphodiesterase 10A(PDE10A)inhibitor.TAK-063 is currently being evaluated in clinical trials for the treatment of schizophrenia.Phosphodiesterase 10A(PDE10A)is a cAMP/cGMP phosphodiesterase highly expressed in medium spiny neurons(MSNs)in the striatum.TAK-063 represents a promising drug for the treatment of schizophrenia with potential for superior safety and tolerability profiles. | price> |
R-C-2830 | Oil soluble MnxFe3-xO4 nanoparticles | The average autocatalytic reaction order of MnxFe3-xO4 nanoparticles increased from 0.48 of pure epoxy to 0.52 of epoxy/MnxFe3-xO4 nanocomposites, because the hydroxyl groups on the surface of nanoparticles participated in the ring opening of epoxides. | price> |
R-R-2830 | Glepaglutide acetate | Glepaglutide (ZP1848) acetate, a long-acting GLP-2 analogue, is a potent GLP-2R agonist. Glepaglutide acetate reduces faecal output and increases intestinal absorption. Glepaglutide acetate alleviates small intestinal inflammation. | price> |
R-C-1131 | SB239063 CAS:193551-21-2 | SB 239063 is a selective p38 MAPK inhibitor(IC50=44 nM for recombinant purified p38α).1 It displays greater than 220-fold selectivity for p38 MAPK over ERK, JNK1,and other kinases.1 SB 239063 has been shown to reduce inflammatory cytokine production in lipopolysaccharide-stimulated human peripheral blood monocytes(IC50s=0.12 and 0.35 µM,respectively for IL-1 and TNF-α)and is neuroprotective following oral administration in a rat model of cerebral focal ischemia. | price> |
R-C-2831 | Mannose/chitosan loaded on liposome surface(90nm) | Long circulating liposomes can inhibit tumor and regulate immunity Chitosan, a natural polymer,has excellent properties such as biological functionality and compatibility,blood compatibility,safety,microbial degradation and so on. | price> |
R-R-2831 | GLP-2(3-33) CAS No.275801-62-2 | GLP-2(3-33)/CAS No.275801-62-2, generated naturally by dipeptidylpeptidase IV (DPPIV), acts as a partial agonist on GLP-2 receptor (EC50=5.8 nM). | price> |
R-C-1132 | BIBX1382 CAS:196612-93-8 | BIBX 1382 is a cell-permeable pyrimidopyrimidine compound that acts as a potent, reversible,ATP-competitive,and highly selective inhibitor of EGFR. | price> |
R-C-2832 | DSPE-NBD | 1,2-distearoyl-sn-glycoro-3-phosphoethanolamine-nitrobenzofurazan is produced by Xi an Ruixi biology.Our company can also produce various customized products. | price> |
R-R-2832 | Glucagon receptor antagonists-3 CAS No.202917-17-7 | Glucagon receptor antagonists-3/CAS No.202917-17-7 is a highly potent glucagon receptor antagonist. | price> |
R-C-1133 | GSKJ1 CAS :1373422-53-7 | GSKJ1 is a selective and potent histone demethylase inhibitor(GSK-J1)that has significant activity(IC50 60 nM for human JmjD3)in vitro and in cells using an ester derivative(GSK-J4:1 µMprice> |
|
R-C-2833 | PLA5K-PEG2K-Heparin nanoparticles | The former is helpful to improve the biocompatibility,targeting and drug loading of nanoparticles,while the latter is mainly used for the targeted transport of proteins and antitumor drugs. | price> |
R-R-2833 | Mazdutide CAS No.2259884-03-0 | Mazdutide (IBI-362; LY-3305677)/CAS No.2259884-03-0 is a long-acting synthetic oxyntomodulin analog. Mazdutide is also a co-agonist of glucagon-like peptide (GLP-1R) and?glucagon receptor?(GCGR). Mazdutide binds human and mouse?GCGR?(Ki: 17.7 nM and 15.9 nM, respectively) and GLP-1R (Ki: 28.6 nM and 25.1 nM, respectively) and stimulates?insulin?secretion from mouse islets (EC50: 5.2 nM). Mazdutide is used in studies of obesity and type 2 diabetes (T2D). | price> |
R-C-1134 | SEP-0372814 CAS:1516895-53-6 | SEP-0372814 is an inhibitor of phosphodiesterase 10A(PDE10A;IC50≤10 nM for the recombinant human enzyme). | price> |
R-C-2834 | PLA5K-PEG2K-Heparin loaded nanoparticles | Poly(L-lactide)is a amphiphilic AB block copolymer,the PEG hydrophilic is capped a maleimidegroup,and the PDLLA hydrophobic block terminates with a hydroxyl group. | price> |
R-R-2834 | L-168049 CAS No.191034-25-0 | L-168049/CAS No.191034-25-0 is a potent, selective, orally active and non-competitive glucagon receptor antagonist with IC50s of 3.7 nM, 63 nM, and 60 nM for human, murine, and canine glucagon receptors, respectively. | price> |
R-C-1135 | BIO-32546 CAS NO. 1548743-66-3 | BIO-32546 is a novel modulator of the activity of the autotaxin(ATX)enzyme. | price> |
R-C-2835 | PLA5K-PEG2K-NH2 nanoparticles | The products of RuixiBiotechCo.Ltd include synthetic phospholipids,high molecular polyethylene glycol derivatives,block copolymers,magnetic nanoparticles,nano gold and nano gold rods,near-infrared fluorescent dyes, reactive fluorescent dyes, fluorescent labeled dextran BSA and streptavidin, protein crosslinking agents,small molecular PEG derivatives, counting chemical products Dendrimers,cyclodextrin derivatives,popular APIs,macrocyclic ligands,fluorescent quantum dots,hyaluronic acid derivatives,graphene or graphene oxide,carbon nanotubes,fullerenes,etc. | price> |
R-R-2835 | Shanzhiside methyl ester CAS No.64421-28-9 | Shanzhiside methy lester/CAS No.64421-28-9 is isolated from lamiophlomis rotata. Shanzhiside methyl ester is a small molecule glucagon-like peptide-1 (GLP-1) receptor agonist and has the ability to induce anti-allodynic tolerance. | price> |
R-C-1136 | PF-562271 CAS :717907-75-0 | PF-562271 Besylate is the benzenesulfonate salt of PF-562271,which is a potent,ATP-competitive,reversible inhibitor of FAK with IC50 of 1.5 nM,~10-fold less potent for Pyk2 than FAK and>100-fold selectivity against other protein kinases,except for some CDKs. | price> |
R-R-2836 | VU0453379 hydrochloride | VU0453379 hydrochloride is a highly selective and central nervous system (CNS) penetrant positive allosteric modulator (PAM) of glucagon-like peptide-1R (GLP-1R) with an EC50 of 1.3 μM. | price> |