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Catalog	name	Description	price
R-R-2891	SKF-83566 CAS No.99295-33-7	SKF-83566/CAS No.99295-33-7 is a potent, blood-brain permeable and orally active D1-like dopamine receptor (D1DR) antagonist and a weaker competitive antagonist at the vascular 5-HT2 receptor (Ki=11 nM). SKF-83566 is a competitive DAT (dopamine transporter) inhibitor with an IC50 of 5.7 μM. SKF-83566 also shows selective inhibition for adenylyl cyclase 2 (AC2) over AC1 and AC5 in the isolated rabbit thoracic aorta.	price>
R-C-1192	RQ-00203078 CAS:1254205-52-1	RQ-00203078 is a highly selective,potent and orally available TRPM8 antagonist (IC50 values are 5.3 and 8.3 nM for rat and human channels respectively), exhibits>350-fold selectivity for TRPM8 over TRPV4,TRPV1 and TRPA1.	price>
R-R-2892	ST034307 CAS No.133406-29-8	ST034307/CAS No.133406-29-8 is a potent and selective adenylyl cyclase 1 (AC1) inhibitor, with IC50 of 2.3 μM.	price>
R-C-1193	Kevetrin HCl	Kevetrin hydrochloride is a small molecule and activator of the tumor suppressor protein p53,with potential antineoplastic activity.	price>
R-R-2893	NKY80 CAS No.299442-43-6	NKY80/CAS No.299442-43-6 is a potent, selective and non-competitive adenylyl cyclase (AC) type V isoform inhibitor with IC50s of 8.3 µM, 132 µM and 1.7 mM for type V, III and II, respectively. NKY80 is a non-nucleoside quinazolinone and regulates the AC catalytic activity in heart and lung tissues.	price>
R-C-1194	LY310762 CAS:192927-92-7	LY310762 is a 5-HT1D antagonist with Ki of 249 nM, having a weaker affinity for 5-HT1B receptor.	price>
R-R-2894	Guanylyl imidodiphosphate lithium CAS No.64564-03-0	Guanylyl imidodiphosphate (Gpp(NH)p) lithium/CAS No.64564-03-0, a non-hydrolyzable GTP analogue, increases adenylate cyclase activity.	price>
R-C-1195	GSK-LSD1 CAS:2102933-95-7	GSK-LSD1 dihydrochloride is a potent,selective and irreversible lysine specific demethylase 1(LSD1)inhibitor with an IC50 of 16 nM.	price>
R-R-2895	TDI-11861 CAS No.2857049-72-8	TDI-11861/CAS No.2857049-72-8 is second-generation soluble Adenylyl Cyclase (sAC, ADCY10) inhibitor with slow dissociation rates. TDI-11861 inhibits sAC cellular with an IC50 value of 5.5 nM.	price>
R-C-1196	ORY-1001 CAS：1431326-61-2	ORY-1001 is an orally active and selective lysine-specific demethylase LSD1/KDM1A inhibitor with IC50 of <20 nM,with high selectivity against related FAD dependent aminoxidases.	price>
R-R-2896	Fipexide hydrochloride CAS No.34161-23-4	Fipexide hydrochloride/CAS No.34161-23-4, a parachloro-phenossiacetic acid derivative, is an orally active nootropic agent. Fipexide hydrochloride reduces striatal adenylate cyclase activity. Fipexide hydrochloride has positive effect on cognitive performance by dopaminergic neurotransmission. Fipexide hydrochloride is used for senile dementia research. Fipexide hydrochloride acts as a chemical inducer in callus formation, shoot regeneration and Agrobacterium infection.	price>
R-C-1197	CPI-268456	CPI-268456 is a ligand of bromodomain-containing protein 4(BRD4).It binds to BRD4(IC5=<0.5 µM in a cell-free assay)and inhibits LPS-induced IL-6 secretion in THP-1 cells(IC50=<0.5 µM).	price>
R-R-2897	Lysipressin acetate CAS No.83968-49-4	Lysipressin (Lysine vasopressin) acetate/CAS No.83968-49-4 is antidiuretic hormone that have been found in pigs and some marsupial families. Lysipressin acetate induces contraction of the rabbit urinary bladder smooth muscle, activate adenylate-cyclase.	price>
R-C-1198	SW-033291 CAS：459147-39-8	SW033291 is a potent and high-affinity inhibitor of 15-PGDH with a Ki of 0.1 nM.SW033291 increases prostaglandin PGE2 levels in bone marrow and other tissues. SW033291 also promotes tissue regeneration.	price>
R-R-2898	9-Cyclopentyladenine monomethanesulfonate CAS No.189639-09-6	9-Cyclopentyladenine monomethylsulfonate (9-CP-Ade mesylate)/CAS No.189639-09-6 is a stable non-competitive adenylate cyclase inhibitor with cell permeable properties.	price>
R-C-1199	IBET762(GSK525762A) CAS ：1260907-17-2	Molibresib(I-BET-762,GSK525762,GSK525762A)is an inhibitor for BET proteins with IC50 of ~35 nM in a cell-free assay,suppresses the production of proinflammatory proteins by macrophages and blocks acute inflammation,highly selective over other bromodomain-containing proteins.	price>
R-R-2899	Zelminemab CAS No.2225850-33-7	Zelminemab (AMG-301)/CAS No.2225850-33-7 is a human monoclonal antibody that inhibits PACAP type I (PAC1) receptor.	price>
R-C-1200	GSK923295 Cytoskeletal Signaling	GSK-923295 is a special,allosteric inhibitor of centromere-associated protein-E (CENP-E)kinesin motor ATPase activity,with Ki of 3.2±0.2 nM and 1.6± 0.1 nM for human and canine,respectively.	price>
R-R-2900	CB-7921220 CAS No.115453-99-1	CB-7921220/CAS No.115453-99-1 is an adenylate cyclase inhibitor.	price>
R-C-1201	JZL-195 CAS:1210004-12-8	JZL195 is a selective and efficacious dual FAAH/MAGL inhibitor with IC50 of 13 nM and 19 nM for mouse brain FAAH and MAGL respectively.	price>

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