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Catalog	name	Description	price
R-C-1177	GS-7340(Tenofovir alafenamide ) CAS：379270-37-8	Tenofovir Alafenamide(GS-7340)is a prodrug of tenofovir,which is a reverse transcriptase inhibitor,used to treat HIV and Hepatitis B.	price>
R-R-2877	PA-8 CAS No.878437-15-1	PA-8/CAS No.878437-15-1 is a potent, selective and orally active PACAP type I (PAC1) receptor antagonist. PA-8 inhibits the phosphorylation of CREB induced by PACAP in PAC1-, but not VPAC1- or VPAC2-receptor. PA-8 also inhibits PACAP-induced cAMP elevation with an IC50 of 2 nM.	price>
R-C-1178	GSK503 CAS：1346572-63-1	GSK503 is a potent and specific inhibitor of EZH2 methyltransferase with Kiapp values of 3 to 27 nM.	price>
R-R-2878	PACAP (6-38), human, ovine, rat TFA	PACAP (6-38), human, ovine, rat TFA is a potent PACAP receptor antagonist with IC50s of 30, 600, and 40 nM for PACAP type I receptor, PACAP type II receptor VIP1, and PACAP type II receptor VIP2, respectively.	price>
R-C-1179	CGI-1746 CAS：910232-84-7	CGI1746 is a small-molecule Btk inhibitor chemotype with a new binding mode that stabilizes an inactive nonphosphorylated enzyme conformation.	price>
R-R-2879	PAC1R antagonist 1 CAS No.2305204-24-2	PAC1R antagonist 1 (compound 3d)/CAS No.2305204-24-2 is a potent and orally active antagonist of PAC1 receptor. PAC1R antagonist 1 can inhibit pituitary adenylate cyclase-activating polypeptide (PACAP)- and nerve injury-induced allodynia.	price>
R-C-1180	Endoxifen CAS：112093-28-4	Endoxifen is a secondary metabolite of tamoxifen.It is a primary metabolite responsible for the effectiveness of tamoxifen in ER-positive breast cancer.	price>
R-R-2880	PACAP (1-27), human, ovine, rat TFA	PACAP (1-27), human, ovine, rat TFA (PACAP 1-27 TFA) is the N-terminal fragment of PACAP-38, and is a potent PACAP receptor antagonist with IC50s of 3 nM, 2 nM and 5 nM for rat PAC1, rat VPAC1 and human VPAC2, respectively.	price>
R-C-1181	D-Luciferin CAS ：2591-17-5	D-Luciferin is a popular bioluminescent substrate of luciferase in the presence of ATP,used in luciferase-based bioluminescence imaging and cell-based high-throughput screening applications.	price>
R-R-2881	PACAP (1-38), amide, Biotin-labeled	PACAP (1-38), amide, Biotin-labeled is a biological active peptide. (Biotin-labeled HY-P0221)	price>
R-C-1182	NS6180	NS6180 is a novel potent and selective KCa3.1 channel inhibitor(IC50=9nM) prevents T-cell activation and inflammation.	price>
R-R-2882	PA-9 CAS No.1436004-46-4	PA-9/CAS No.1436004-46-4 is a pituitary adenylate cyclase-activating polypeptide (PACAP) type I (PAC1) receptor antagonist. PA-9 dose dependently inhibits PACAP-induced cAMP elevation with an IC50 of 5.6 nM. PA-9 can be used for the research of neuropathic and/or inflammatory pain.	price>
R-C-1183	Loxiglumide CAS:107097-80-3	Loxiglumide is a potent,orally active,and selective CCK-A receptor antagonist which stimulates calorie intake and hunger feelings in humans.Loxiglumide inhibits pancreatic secretion of digestive enzymes,and also blocks CCK-induced gastric secretions and emptying.Intravenous administration of loxiglumide antagonized the CCK-induced reduction of gastric emptying in rats,acceleration of intestinal transport in mice,increase in ileal motility in rabbits, gallbladder contraction in guinea pigs and acceleration of gallbladder emptying in mice.	price>
R-R-2883	(Tyr36)-pTH-Related Protein (1-36) (human, mouse, rat) CAS No.213779-11-4	(Tyr36)-pTH-Related Protein (1-36) (human, mouse, rat)/CAS No.213779-11-4 is a peptide and can be used as a parathyroid hormone (PTH) receptor ligand.	price>
R-C-1184	BD1047.2HBr CAS 138356-21-5	BD-1047 hydrobromide,a selective functional antagonist of sigma receptors,has antipsychotic activity in animal models predictive of efficacy in schizophrenia.	price>
R-R-2884	Human PTHrP-(1-36) CAS No.172867-62-8	Human PTHrP-(1-36)/CAS No.172867-62-8 is a secretory form of PTHrP with anticalciuric effects. Human PTHrP-(1-36) enhances beta cell function and proliferation. Human PTHrP-(1-36) can be used in the research of humoral hypercalcemia of malignancy (HHM) and hyperparathyroidism.	price>
R-C-1185	Evacetrapib (LY2484595) CAS No. 1186486-62-3	Evacetrapib is a potent and selective of CETP inhibitor,which inhibits human recombinant CETP protein(IC50 5.5 nM)and CETP activity in human plasma(IC50 36 nM)in vitro.	price>
R-R-2885	Secretin (33-59), rat TFA	Secretin (33-59), rat (TFA) is a 27-aa peptide, which acts on secretin receptor, and enhances the secretion of bicarbonate, enzymes, and K+ from the pancreas.	price>
R-C-1186	TAE226 (NVP-TAE226) CAS:761437-28-9	NVP-TAE 226(TAE226)is a potent and ATP-competitive dual FAK and IGF-1R inhibitor with IC50s of 5.5 nM and 140 nM,respectively.NVP-TAE 226(TAE226) also effectively inhibits Pyk2 and insulin receptor(InsR)with IC50s of 3.5 nM and 44 nM,respectively.	price>
R-R-2886	NKH477 CAS No.138605-00-2	NKH477 (Colforsin dapropate hydrochloride)/CAS No.138605-00-2 directly activates the catalytic unit of adenylate cyclase and increases intracellular cAMP. NKH477 is a forskolin derivative that improves cardiac failure mainly through its beneficial effects on diastolic cardiac function. NKH477 exerts an antiproliferative effect in vivo with an altered cytokine profile to inhibit the acute rejection of rat orthotopic lung allografts.	price>

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