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R-C-1648 Miransertib (ARQ-092) CAS:1313881-70-7 Miransertib(ARQ-092)is a potent,selective and orally bioavailable allosteric inhibitor of Akt with IC50s of 2.7nM,14 nM and 8.1nM for Akt1,Akt2,Akt3. price>
R-R-3348 SB-200646A CAS No.143797-62-0 SB-200646A/CAS No.143797-62-0 is the first selective 5-HT2B/2C over 5-HT2A receptor antagonist with pKi values of 7.5, 6.9 and 5.2 for 5-HT2B, 5-HT2C and 5-HT2A, respectively. SB-200646A is orally active and has electrophysiological and anxiolytic properties in vivo. price>
R-R-3349 PU02 CAS No.313984-77-9 PU02/CAS No.313984-77-9, a derivative of 6-MP (HY-13677), is a negative allosteric modulator (NAM) of 5-HT3 receptor, with IC50 values of 0.36 and 0.73 μM in HEK293 cells transfected with human 5-HT3A and 5-HT3AB receptors respectively. price>
R-C-1649 SKF96365.HCl CAS:130495-35-1 SKF-96365 hydrochloride is a potent TRP channel blocker and a store-operated Ca2+ entry(SOCE)inhibitor.SKF-96365 hydrochloride significantly inhibits hERG, hKCNQ1/hKCNE1,hKir2.1 and hKv4.3 current,and significantly prolongs the QTc interval in isolated guinea pig hearts.SKF-96365 hydrochloride exhibits potent anti-neoplastic activity by inducing cell-cycle arrest and apoptosis in colorectal cancer cells. price>
R-C-1650 AR-M1000390 HCl  CAS:209808-47-9  AR-M1000390(ARM-390)is a nonpeptidic δ receptor selective agonist. price>
R-R-3350 Alniditan dihydrochloride CAS No.155428-00-5 Alniditan (Alnitidan) dihydrochloride/CAS No.155428-00-5 is a potent 5-HT1B and 5-HT1D receptors agonist, with IC50s of 1.7 nM and 1.3 nM for h5-HT1B and h5-HT1D receptors in HEK 293 cells, respectively. Alniditan dihydrochloride has migraine-preventive effects. price>
R-C-1651 nicainoprol CAS:76252-06-7 Nicainoprol is a fast-sodium-channel blocking drug,which is a potent antiarrhythmic agent. price>
R-R-3351 Tedatioxetine hydrobromide CAS No.960151-65-9 Tedatioxetine (Lu AA24530) hydrobromide/CAS No.960151-65-9 acts as a serotonin and norepinephrine (NE)-preferring triple reuptake inhibitor (TRI) and 5-HT2A, 5-HT2C, 5-HT3 and α1A-adrenergic receptor antagonist. price>
R-C-1652 DAA1106 CAS:220551-92-8 DAA1106 is a potent and selective ligand for peripheral benzodiazepine receptor (PBR),as a potent and selective agonist at the peripheral benzodiazepine receptor. price>
R-R-3352 Naluzotan CAS No.740873-06-7 Naluzotan/CAS No.740873-06-7 is a novel, potent, and selective amidosulfonamide 5-HT1A agonist with IC50 and Ki of appr 20 nM and 5.1 nM, used for the treatment of anxiety and depression; Also a weak hERG K+ channel blocker, with IC50 of 3800 nM. price>
R-C-1653 Eptapirone (F11440) CAS:179756-58-2 Eptapirone(F11440)is a potent,selective,high efficacy 5-HT1A receptor agonist with marked anxiolytic and antidepressant potential. price>
R-R-3353 Velusetrag hydrochloride CAS No.866933-51-9 Velusetrag (TD-5108) hydrochloride/CAS No.866933-51-9 is an orally active, potent and selective agonist of serotonin 5-HT4 receptor (5-HT4R), with a pKi of 7.7. Velusetrag hydrochloride exhibits no affinity (Ki>10 μM) for 5-HT2A and 5-HT2B receptors. price>
R-C-1654 Orexin 2 Receptor Agonist CAS:1796565-52-0 Orexin 2 Receptor Agonist is a potent(EC50 on OX2R is 23nM)and OX2R-selective (OX1R/OX2R EC50 ratio is 70) agonist. price>
R-R-3354 Aripiprazole-d8 CAS No.1089115-06-9 Aripiprazole-d8/CAS No.1089115-06-9 is the deuterium labeled Aripiprazole, which is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM. price>
R-C-1655 piperoxan.HCl CAS: 135-87-5 Piperoxan hydrochloride(Benodaine,Fourneau 933,F933,DL-Piperoxan)is an antagonist of α2(alpha 2)adrenoceptor. price>
R-M-G25 Carbon Nanotube Aerogel Carbon nanotube Aerogel/Carbon nanotubes(CNT) Aerogel/CNT Aerogel is a kind of carbon nanotube with dispersion properties. This paper prepared carbon nanotube aerogel through independent research and development of experimental equipment, and prepared carbon nanotube aerogel/natural rubber composite through traditional processes. Material, the mechanical properties and thermal conductivity of the composite material were studied. The results proved that the tensile strength, tear strength and thermal conductivity of the composite material were improved by 47%, 52% and 49.9 respectively compared with the carbon black/natural rubber composite material. %, while revealing the good dispersion properties of carbon nanotube airgel and its broad application prospects. price>
R-C-1656 pipequaline CAS:77472-98-1 Pipequaline(PK 8165)is a partial benzodiazepine receptor agonist with anxiolytic activity. price>
R-M-G26 La2O3-doped bulk alumina aerogel La2O3 doped bulk alumina aerogels/Lanthanum oxide doped bulk alumina aerogels/La2O3-doped bulk Al2O3 aerogel/Lanthanum oxide doped bulk Al2O3 aerogels with different La2O3 contents are prepared by using aluminum tri-sec-butoxide as precursor via sol-gel route combined with acetone-aniline in situ water formation (ISWF) method, followed by supercritical fluid drying. The effect of La2O3 on microstructure and thermal stability of alumina aerogels is investigated by SEM, TEM, XRD and N2 adsorption. The results show that the morphology of alumina aerogels changes from sphere like accumulated to notably sheet like stacked with the doping of La2O3. An appropriate amount of La2O3 doping can enhance the specific surface area of alumina aerogels, and the 9 mol% La2O3 doping aerogels has the largest specific surface area. In addition, the alumina crystal growth and phase transition of the aerogels upon heat treatment are effectively inhibited by La2O3 doping, which significantly improves the thermal stability of the aerogels. After heat treatment at 1200℃ for 2h, the phase of 9 mol% La2O3 doped alumina aerogel remains in the θ-Al2O3 while that of undoped one is a-Al2O3, and the specific surface area of 9 mol% La2O3 doped alumina aerogel is 86.5 m2/g which is higher than the undoped one (46 m2/g). price>
R-C-1657 nifenalol.HCL CAS# 5704-60-9  Nifenalol(INPEA)hydrochloride is an antagonist of beta-adrenergic receptor. price>
R-AC-0001 Nanocellulose-based composite aerogel (CSP-AG) Nanocellulose-based composite aerogels (CSP-AG) were prepared using carboxylated cellulose nanofibers (CCNF), silane coupling agent (KH560) and polyethylenimine (PEI) as raw materials. By regulating CCNF, KH560 and Different CSP-AGs were prepared by the ratio between PEI. price>