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Catalog	name	Description	price
R-C-1678	Fosaprepitant dimeglumine CAS：265121-04-8	Fosaprepitant dimeglumine(MK-0517)is a prodrug of Aprepitant(HY-10052). Fosaprepitant dimeglumine is a neurokinin-1 receptor antagonist,which is development for the prevention of chemotherapy-induced nausea and vomiting (CINV).	price>
R-R-3378	Revexepride CAS No.219984-49-3	Revexepride/CAS No.219984-49-3 is a highly selective 5-HT4 receptor agonist, and a potential inducer of CYP3A4 enzyme, used for the treatment of gastroesophageal reflux disease.	price>
R-C-1679	Tebipenem pivoxil CAS：161715-24-8	Tebipenem pivoxil(ME1211)SPR994 and TBM-PI,is a novel oral carbapenem antibiotic.TBM-PI is a promising antibiotic for the treatment of acute otitis media.Tebipenem pivoxil displays an excellent antibacterial activity against a variety of pathogenic bacteria in vitro.	price>
R-R-3379	Relenopride hydrochloride CAS No.1221416-42-7	Relenopride (YKP10811) hydrochloride/CAS No.1221416-42-7 is a specific and selective 5-HT4 receptor agonist (Ki=4.96 nM). Relenopride hydrochloride has 120-fold and 6-fold lower affinity, respectively, for 5-HT2A (Ki=600 nM) and 5-HT2B receptors (Ki=31 nM) than for 5-HT4. Relenopride hydrochloride increases gastrointestinal (GI) motility.	price>
R-C-1680	Carteolol hydrochloride CAS：51781-21-6	Carteolol hydrochloride(OPC-1085 hydrochloride)is a non-selective beta blocker used to treat glaucoma.	price>
R-R-3380	TC-2153 CAS No.1381769-23-8	TC-2153/CAS No.1381769-23-8 is a selective inhibitor of striatal-enriched protein tyrosine phosphatase (STEP), with psychotropic activity and low acute toxicity. TC-2153 increases the expression of brain-derived neurotropic factor (BDNF) in the brain. And it decreases MAOA and 5-HT1A receptors mRNA level in midbrain. TC-2153 also inhibits 5-HT2A receptor-mediated signaling.	price>
R-C-1681	1400W dihydrochloride CAS：214358-33-5	1400W dihydrochloride is a potent and selective inhibitor of human inducible NO synthase with Ki values of 7nM.	price>
R-R-3381	(R)-Praziquantel-d11 CAS No.1399880-38-6	(R)-Praziquantel-d11/CAS No.1399880-38-6 is the deuterium labeled (R)-Praziquantel. (R)-Praziquantel, the active enantiomer of Praziquantel, is a partial agonist of the human 5-HT2B receptor. (R)-Praziquantel acts as an antischistosomal eutomer.	price>
R-C-1682	SQ22536 CAS：17318-31-9	SQ22536(9-(tetrahydrofuran-2-yl)-9h-purin-6-amine)is an inhibitor of adenylyl cyclase with an IC50 of 1.4μM.It can inhibit PGE1-stimulated increases in cAMP levels in intact human platelets.	price>
R-R-3382	Clozapine-d8 CAS No.1185053-50-2	Clozapine-d8/CAS No.1185053-50-2 is the deuterium labeled Clozapine. Clozapine is an antipsychotic used for the research of schizophrenia. Clozapine has high affinity for a number of neuroreceptors.	price>
R-C-1683	LY2801653 CAS：1206799-15-6	Merestinib(LY2801653)is a type-II ATP competitive,slow-off inhibitor of Met(c-Met)tyrosine kinase with a dissociation constant(Ki)of 2 nM, a pharmacodynamic residence time(Koff)of 0.00132 min(-1)and t1/2 of 525 min.Merestinib (LY2801653) also inhibits MST1R,AXL,ROS1,MKNK1/2, FLT3,MERTK,DDR1 and DDR2 with IC50 of 11 nM,2nM,23nM,7nM,7nM,10 nM,0.1nM and 7nM,respectively.	price>
R-R-3383	Ipsapirone CAS No.95847-70-4	Ipsapirone (TVX Q 7821)/CAS No.95847-70-4 is an anxiolytic compound and a 5-HT1A receptor partial agonist. Ipsapirone (TVX Q 7821) also exhibits 5-HT1A receptor antagonistic effect, and only at high doses it can also produce an inhibitory effect on 5-HT2 and the α1-adrenergic function.	price>
R-C-1684	CRT0066101 2HCL CAS：1883545-60-5	CRT0066101 dihydrochloride is a small molecule PKD family specific inhibitor which specifically blocks PKD1/2 activity and does not suppress PKCα/PKCβ/PKCε activity in multiple.	price>
R-R-3384	Iprindole CAS No.5560-72-5	Iprindole/CAS No.5560-72-5, a tricyclic indole antidepressant, is a weak inhibitor of the uptake of noradrenaline and 5-HT.	price>
R-C-1685	KR-33494 CAS:1021497-97-1	KR-33494 is a fluorescent-tagged and biotin-tagged probe of a potent inhibitor for Fas-mediated cell death(FAF1).	price>
R-R-3385	cis-(Z)-Flupentixol dihydrochloride CAS No.51529-01-2	cis-(Z)-Flupentixol dihydrochloride/CAS No.51529-01-2 is a potent and selective DA D1/D2 receptor antagonist, with Ki values of 0.38 nM and 7 nM for D2 receptor and 5-HT2A, respectively.	price>
R-C-1686	MK 0557 CAS:328232-95-7	MK-0557 is a highly selective,orally administered neuropeptide NPY5R antagonist,could limit weight regain after very-low-calorie diet(VLCD)-induced weight loss.Neuropeptide Y(NPY)is a potent orexigenic neuropeptide,and antagonism of NPY Y1 and NPY Y5 receptors(NPYxR)is considered a potentially important anti-obesity drug target.	price>
R-R-3386	Prucalopride-13C,d3 CAS No.2140306-00-7	Prucalopride-13C,d3/CAS No.2140306-00-7 is the 13C- and deuterium labeled Prucalopride.	price>
R-C-1687	NMS-P118 CAS：1262417-51-5	NMS-P118 is a potent,orally available,and highly selective PARP-1 inhibitor endowed with excellent ADME and pharmacokinetic profiles,showing 150-fold selectivity for PARP-1 over PARP-2(Kd 0.009μM vs 1.3μM,respectively).	price>
R-R-3387	LY 344864 racemate CAS No.186543-64-6	LY 344864 racemate/CAS No.186543-64-6 is a 5-HT1F receptor agonist extracted from patent US 5708187 A.	price>

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