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Catalog	name	Description	price
R-C-1837	ZINC00881524 (ROCK inhibitor) CAS:557782-81-7	ZINC00881524 is a potent and selective ROCK inhibitor.Clinically,inhibition of ROCK pathway is believed to contribute to some of the cardiovascular benefits of statin therapy that are independent of lipid lowering(ie,pleiotropic effects).	price>
R-R-3537	LAS101057 CAS No.925676-48-8	LAS101057/CAS No.925676-48-8 is a potent, selective, and orally efficacious A2B receptor antagonist.	price>
R-C-1838	VH298 CAS:2097381-85-4	VH298 is a potent VHL(Von Hippel-Lindau,the E3 ligase)inhibitor that stabilizes HIF-α.VH298 blocks the VHL:HIF-α interaction with Kd of 90 nM in isothermal titration calorimetry(ITC)and 80 nM in a competitive fluorescence polarization assay.VH-298 can be used in PROTAC technology.	price>
R-R-3538	Tozadenant CAS No.870070-55-6	Tozadenant/CAS No.870070-55-6 is an adenosine A2A receptor antagonist, with Ki of 11.5 nM on human A2A and 6 nM on rhesus A2A.	price>
R-C-1839	VCMMAE CAS:646502-53-6	VcMMAE(mc-vc-PAB-MMAE),a MMAE derivative with valine-citrulline(Vc)linker,is an antibody-drug conjugate(ADC)with potent antitumor activity.MMAE is a synthetic antineoplastic agent and can be efficiently released from VcMMAE in vitro and exert cytotoxic activity.	price>
R-R-3539	N6-Ethyladenosine CAS No.14357-08-5	N6-Ethyladenosine/CAS No.14357-08-5 is an adenosine derivative, acts as a Adenosine receptor agonist, with Kis of 4.9 and 4.7 nM for hA1AR and hA3AR, respectively.	price>
R-C-1840	SC-560 CAS：188817-13-2	SC-560 is a highly selective COX-1 inhibitor with IC50 of 9nM,compared with the IC50 of 6.3μM for COX-2,nearly 1,000-fold higher than with COX-1.	price>
R-R-3540	N6-(2-Phenylethyl)adenosine CAS No.20125-39-7	N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine)/CAS No.20125-39-7, an adenosine derivative, is a potent adenosine receptors (AR) agonist with Ki values of 11.8 nM, 30.1 nM, 0.63 nM for rat A1AR, human A1AR and hA3AR, respectively.	price>
R-C-1841	Belizatinib (TSR011) CAS：1357920-84-3	Belizatinib is an oral,dual,potent inhibitor of ALK and TRKA,TRKB,and TRKC, with IC50 of 0.7 nM for wild-type recombinant ALK kinase.	price>
R-R-3541	DPTN dihydrochloride CAS No.325767-87-1	DPTN/CAS No.325767-87-1 is a potent and selective human, mouse, and rat A3AR antagonist with Ki values of 1.65, 9.61, and 8.53 nM, respectively.	price>
R-C-1842	H3B-6527 CAS：1702259-66-2	H3B-6527 is a highly selective covalent FGFR4 inhibitor with an IC50 value of <1.2 nM and at least 250-fold selectivity over FGFR1-3(IC50 values of 320,1,290 and 1,060nM respectively).	price>
R-R-3542	M1069	M1069 is a selective and orall active, dual A2A/A2B adenosine receptor antagonist with a selectivity of >100 fold against the A1 and A3 receptors. M1069 counteracts immune-suppressive mechanisms of adenosine, and exhibits anti-tumor activity.	price>
R-C-1843	Alexa Fluor 594 meta-isomer/CAS No.:295348-87-7	Alexa Fluor 594 meta-isomer/CAS No.:295348-87-7 is a fluorescent dye known for its bright red fluorescence. It is commonly used in various biological and chemical applications due to its high photostability and water solubility. This compound is particularly valuable in imaging and flow cytometry, where it provides stable signal generation .	price>
R-R-3543	MIPS521 CAS No.1146188-19-3	MIPS521/CAS No.1146188-19-3 is a positive allosteric modulator of adenosine A1 receptor (A1AR). MIPS521 also has a lower A1R allosteric affinity (pKB=4.95; KB=11 μM). MIPS521 exhibits pain-relieving effects in vivo through modulation of the increased levels of endogenous adenosine.	price>
R-C-1844	MBX-8025 (seladelpar) CAS: 851528-79-5	Seladelpar(MBX-8025)is an orally active,potent(50% effect concentration EC50 2nM),and specific PPAR-δagonist.	price>
R-R-3544	N-[(4-Aminophenyl)methyl]adenosine CAS No.95523-13-0	N-[(4-Aminophenyl)methyl]adenosine/CAS No.95523-13-0 is a adenosine receptor inhibitor, with Ki of 29 nM for Rat ecto-5-Nucleotidase.	price>
R-R-3545	Trabodenoson CAS No.871108-05-3	Trabodenoson (INO-8875)/CAS No.871108-05-3, an adenosine mimetic, is a highly selective Adenosine A1 receptor agonist. Trabodenoson (INO-8875) is used in the study for Primary Open-Angle Glaucoma.	price>
R-C-1845	SGI7079 CAS:1239875-86-5	SGI-7079,a novel selective Axl inhibitor with an IC50 of 58 nM in vitro, inhibits tumor growth in a dose dependent manner and is a potential therapeutic target for overcoming EGFR inhibitor resistance.	price>
R-C-1846	BI-882370 CAS:1392429-79-6	BI-882370 is a potent and selective RAF kinase inhibitor that binds to the ATP binding site of the kinase positioned in the DFG-out(inactive)conformation of the BRAF kinase.BI-882370(BI 882370)inhibits the oncogenic BRAFV600E-mutant,the WT BRAF and CRAF kinases with IC50s of 0.4,0.8,and 0.6nM,respectively.BI-882370 also inhibits SRC family kinases.	price>
R-R-3546	Adenosine amine congener CAS No.96760-69-9	Adenosine amine congener (ADAC)/CAS No.96760-69-9 is a selective A1 adenosine receptor agonist, can ameliorate noise- and Cisplatin-induced cochlear injury. Adenosine amine congener also has neuroprotective effects.	price>

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