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Catalog	name	Description	price
R-C-2098	fulacimstat(BAY1142524) CAS： 1488354-15-9	Fulacimstat is an orally available chymase inhibitor,with IC50s of 4,3nM for human and hamster chymase enzyme,respectively.	price>
R-R-3798	Clorprenaline hydrochloride CAS No.6933-90-0	Clorprenaline hydrochloride/CAS No.6933-90-0 is a β2-adrenergic receptor agonist that is implicated in bronchial expansion. Clorprenaline has the potential for asthma research.	price>
R-C-2099	(-)-(S)-B973B CAS：2244989-34-0	(-)-(S)-B-973B is a potent allosteric agonist and positive allosteric modulator of α7 nAChR,with antinociceptive activity.	price>
R-R-3799	Guanadrel CAS No.40580-59-4	Guanadrel/CAS No.40580-59-4 is an orally active postganglionic adrenergic inhibitor of spiroketal. Guanadre can be used in anti-hypertensive studies.	price>
R-C-2100	CT-1812 CAS：1802632-22-9	CT-1812 is a first-in-class,orally available sigma-2/PGRMC1 antagonist(alpha beta oligomer receptor antagonist),is being developed by Cognition.sCT-1812 is a novel therapeutic candidate for Alzheimer is disease.	price>
R-R-3800	LY377604 CAS No.204592-94-9	LY377604/CAS No.204592-94-9 is a human β3-adrenergic receptor agonist with an EC50 of 2.4 nM and also a β1- and β2-adrenergic receptor antagonist.	price>
R-C-2101	BAY-545 CAS：1699717-32-2	BAY-545 is a potent and selective A2B adenosine receptor antagonist, with an IC50 of 59 nM. BAY-545 also exhibits IC50s of 66,400,280 nM for human, mouse,rat A2B adenosine receptor in cells,respectively,and a Ki of 97nM for human A2B adenosine receptor,with more selectivity over A1,A2A,and A3 adenosine receptor.	price>
R-R-3801	Apraclonidine hydrochloride CAS No.73218-79-8	Apraclonidine hydrochloride (ALO 2145)/CAS No.73218-79-8, a selective α2 and weak α1 receptor agonist activity, effectively lowers intraocular pressure (IOP) in human eyes. Apraclonidine hydrochloride is a topical ophthalmic solution and has the ability to elevate the eye lid.	price>
R-C-2102	Ingliforib CAS：186392-65-4	Ingliforib is a glycogen phosphorylase inhibitor,with IC50s of 52,352 and 150nM for liver,muscle and brain glycogen phosphorylase,and has cardioprotective activity.	price>
R-R-3802	Tizanidine hydrochloride CAS No.64461-82-1	Tizanidine hydrochloride/CAS No.64461-82-1 is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.	price>
R-C-2103	Batefenterol CAS：743461-65-6	Batefenterol(GSK961081;TD-5959)is a novel muscarinic receptor antagonist and β2-adrenoceptor agonist;displays high affinity for hM2,hM3 muscarinic and hβ2-adrenoceptor with Ki values of 1.4,1.3 and 3.7nM,respectively.	price>
R-R-3803	Lofexidine hydrochloride CAS No.21498-08-8	Lofexidine (hydrochloride)/CAS No.21498-08-8 is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal.	price>
R-C-2104	BAR 502 CAS：1612191-86-2	BAR502 is a dual FXR and GPBAR1 agonist.BAR-502 promotes browning of white adipose tissue and reverses liver steatosis and fibrosis.BAR502 protects against liver damage caused by HFD by promoting the browning of adipose tissue.	price>
R-R-3804	Ritodrine hydrochloride CAS No.23239-51-2	Ritodrine (DU21220) hydrochloride/CAS No.23239-51-2 is a β-adrenergic agonist, also an effective smooth muscle and uterine relaxant. Ritodrine hydrochloride prolongs contraction interval, can be used for researching arrest premature labor.	price>
R-C-2105	BAR 501 CAS： 1632118-69-4	BAR501 is a potent and selective G protein-coupled bile acid receptor 1(GPBAR1, GPCR19,TGR5)agonist that effectively transactivates GPBAR1 in HEK293 cells overexpressing a CRE along with GPBAR1 with EC50 of 1μM.	price>
R-R-3805	Indoramin CAS No.26844-12-2	Indoramin/CAS No.26844-12-2 is an orally active antihypertensive agent. Indoramin is also selective for the α1A-adrenoceptor.	price>
R-C-2106	GSK3117391 CAS：1018673-42-1	GSK3117391(GSK3117391A)and HDAC-IN-3,is a potent HDAC inhibitor for treating chronic inflammatory disorders.	price>
R-R-3806	Bucindolol CAS No.71119-11-4	Bucindolol/CAS No.71119-11-4 is a β1-adrenergic receptor blocker, with intrinsic sympathomimetic activity, used in the research of heart failure.	price>
R-C-2107	PZ-2891 CAS：2170608-82-7	PZ-2891 is an orally bioavailable,brain penetrant pantothenate kinase (PANK)modulator.PZ-2891 act as an orthosteric inhibitor at high concentrations and an allosteric activator at lower sub-saturating concentrations.PZ-2891 inhibits human pantothenate kinases PANK1β,PANK2,and PANK3 with IC50s of 40.2 nM,0.7nM and 1.3nM,respectively.	price>
R-R-3807	(R)-Terazosin CAS No.109351-34-0	(R)-Terazosin/CAS No.109351-34-0 is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent α1-adrenoceptor antagonist with Ki values of 6.51 nM, 1.01 nM and 1.97 nM for α1a, α1b and α1d-adrenoceptor, respectively.	price>

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