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Catalog	name	Description	price
R-C-2249	AT13148 CAS： 1056901-62-2	AT13148 is an orally active and ATP-competitive,multi-AGC kinase inhibitor with IC50s of 38nM/402 nM/50nM,8nM,3nM,and 6nM/4nM for Akt1/2/3,p70S6K,PKA，and ROCKI/II,respectively.	price>
R-R-3949	3-Ethylrhodanine CAS :7648-01-3	3-Ethylrhodanine/3-Ethyl-2-Thioxo-1,3-Thiazolan-4-One/CAS :7648-01-3 is a merocyanine dye that has an ethyl group attached to the rhodanine ring. It is produced by condensation of 2-bromo-3-nitrobenzoic acid with carbon disulfide in the presence of an acceptor molecule. This chemical process can be carried out at room temperature and produces high yields. 3-Ethylrhodanine has been shown to have a variety of electrochemical applications, such as nature, devices, morphology and efficiencies. The red shift observed in this dye was found to be due to the alkyl substituents on the carbon atoms adjacent to the nitrogen atom in the rhodanine ring. We can mass produce (kg level), process scaling up, pilot supply, raw material supply, and intermediate production. Our production technology is mature and more cost-effective. Feel free to inquire at any time.	price>
R-C-2250	Cinobufagin CAS：470-37-1	Cinobufagin(Cinobufagine),an active ingredient of Venenum Bufonis,inhibits tumor development.Cinobufagin increases ATM and Chk2 and decreases CDC25C,CDK1,and cyclin B.Cinobufagin inhibits PI3K,AKT and Bcl-2 while increases levels of cleaved caspase-9 and caspase-3. Thus,Cinobufagin induces cell cycle arrest at the G2/M phase and apoptosis.	price>
R-R-3950	Midodrine-d6 hydrochloride CAS No.1188265-43-1	Midodrine-d6 (hydrochloride)/CAS No.1188265-43-1 is deuterium labeled Midodrine, which is a vasopressor/antihypotensive agent.	price>
R-R-3951	Vilanterol-d4 trifenatate CAS No.2021249-10-3	Vilanterol-d4 (trifenatate)/CAS No.2021249-10-3 is deuterium labeled Vilanterol (trifenatate). Vilanterol trifenatate (GW642444 trifenatate) is a long-acting β2-adrenoceptor (β2-AR) agonist with inherent 24-hour activity. The pEC50s for β2-AR, β1-AR and β3-AR are 10.37, 6.98 and 7.36, respectively.	price>
R-R-3952	Oxprenolol-d7 CAS No.1189805-10-4	Oxprenolol-d7/CAS No.1189805-10-4 is the deuterium labeled Oxprenolol. Oxprenolol (Ba 39089 free base) is an orally bioavailable β-adrenergic receptor (β-AR) antagonist with a Ki of 7.10 nM in a radioligand binding assay using rat heart muscle.	price>
R-R-3953	Brimonidine-d4 CAS No.1184971-51-4	Brimonidine-d4/CAS No.1184971-51-4 is the deuterium labeled Brimonidine. Brimonidine (UK 14304) is a full α2-adrenergic receptor (α2-AR) agonist.	price>
R-R-3954	Benoxathian hydrochloride CAS No.92642-97-2	Benoxathian hydrochloride/CAS No.92642-97-2 is a potent α1 adrenoceptor antagonist, can be used for researching anorexia.	price>
R-R-3955	Brimonidine-d4 D-tartrate CAS No.1316758-27-6	Brimonidine-d4 (D-tartrate)/CAS No.1316758-27-6 is the deuterium labeled Brimonidine D-tartrate.	price>
R-R-3956	Tetrahydrozoline-d4 hydrochloride CAS No.1246814-66-3	Tetrahydrozoline-d4 (hydrochloride)/CAS No.1246814-66-3 is the deuterium labeled Tetrahydrozoline hydrochloride. Tetrahydrozoline hydrochloride (Tetryzoline hydrochloride), a derivative of imidazoline, is an α-adrenergic agonist that causes vasoconstriction. Tetrahydrozoline hydrochloride is widely used for the research of nasal congestion and conjunctival congestion.	price>
R-R-3957	ST91 CAS No.4749-61-5	ST91/CAS No.4749-61-5 is a α2-adrenoceptor (α2AR) agonist. ST91 activates both α2AAR and non-α2AAR subtypes to produce spinal antinociception.	price>
R-R-3958	Octopamine-d4 hydrochloride CAS No.1219803-62-9	Octopamine-d4 (hydrochloride)/CAS No.1219803-62-9 is the deuterium labeled Octopamine hydrochloride. Octopamine ((±)-p-Octopamine) hydrochloride, a biogenic monoamine structurally related to noradrenaline, acts as a neurohormone, a neuromodulator and a neurotransmitter in invertebrates. Octopamine hydrochloride can stimulate alpha2-adrenoceptors (ARs) in Chinese hamster ovary cells transfected with human alpha2-ARs. Octopamine hydrochloride increased glycogenolysis, glycolysis, oxygen uptake, gluconeogenesis and the portal perfusion pressure.	price>
R-R-3959	Amitriptyline hydrochloride (Standard) CAS No.549-18-8	Amitriptyline (hydrochloride) (Standard)/CAS No.549-18-8 is the analytical standard of Amitriptyline (hydrochloride). This product is intended for research and analytical applications. Amitriptyline hydrochloride is an inhibitor of serotonin reuptake transporter (SERT) and noradrenaline reuptake transporter (NET), with Kis of 3.45 nM and 13.3 nM for human SERT and NET, respectively. Amitriptyline hydrochloride also weakly binds to dopamine reuptake transporter (DAT) with a Ki of 2.58 μM. Amitriptyline hydrochloride also inhibits adrenergic, muscarinic, histamine and 5-HT receptors. Amitriptyline hydrochloride is a TrkA and TrkB receptors agonist with potent neurotrophic activity. Amitriptyline hydrochloride has antidepressant activity.	price>
R-R-3960	Butyryltimolol CAS No.106351-79-5	Butyryltimolol/CAS No.106351-79-5, an effective precursor of Timolol, improves the corneal penetration of Timolol. Butyryltimolol is a β-adrenergic blocker.	price>
R-R-3961	Prazosin-d8 hydrochloride CAS No.1189508-34-6	Prazosin-d8 hydrochloride/CAS No.1189508-34-6 is the deuterium labeled Prazosin hydrochloride. Prazosin hydrochloride is an alpha-adrenergic blocker.	price>
R-R-3962	Piribedil-d8 CAS No.1398044-45-5	Piribedil-d8/CAS No.1398044-45-5 is the deuterium labeled Piribedil, which is an antiparkinsonian agent.	price>
R-R-3963	Carazolol-d7 CAS No.1173021-02-7	Carazolol-d7/CAS No.1173021-02-7 is the deuterium labeled Carazolol.	price>
R-R-3964	Mirtazapine-d4 CAS No.1215898-55-7	Mirtazapine-d4/CAS No.1215898-55-7 is deuterium labeled Mirtazapine. Mirtazapine (Org3770) is a potent and orally active noradrenergic and specific serotonergic antidepressant (NaSSA) agent. Mirtazapine is also a 5-HT2, 5-HT3, histamine H1 receptor and α2-adrenoceptor antagonist with pKi values of 8.05, 8.1, 9.3 and 6.95, respectively.	price>
R-C-2265	Ribociclib hydrochloride CAS：1211443-80-9	Ribociclib hydrochloride(LEE011 hydrochloride)is a highly specific CDK4/6 inhibitor with IC50 values of 10nM and 39nM,respectively,and is over 1,000-fold less potent against the cyclin B/CDK1 complex.	price>
R-R-3965	Clorprenaline-d6 CAS No.1648796-40-0	Clorprenaline-d6/CAS No.1648796-40-0 is the deuterium labeled Clorprenaline.	price>

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