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Catalog	name	Description	price
R-C-2420	Dexmedetomidine CAS:113775-47-6	Dexmedetomidine is notable for its ability to provide sedation without risk of respiratory depression(unlike other commonly used sedatives such as propofol, fentanyl,and midazolam)and can provide cooperative or semi-arousable sedation.	price>
R-R-4120	BML-190 CAS No.2854-32-2	BML-190(IMMA)/CAS No.2854-32-2 is a potent and selective CB2 receptor ligand (Ki values are 435 nM and > 2 μM for CB2 and CB1 respectively).	price>
R-C-2421	Pimethixene maleate CAS:13187-06-9	Pimethixene(Pimetixene)maleate,an antihistamine,anntimigraine agent and antiserotonergic compound,is a highly potent antagonist of a broad range of monoamine receptors,including a variety of serotonin receptors.	price>
R-R-4121	Auriculasin CAS No.60297-37-2	Auriculasin/CAS No.60297-37-2 is a nature product isolated from Limonium leptophyllum. Auriculasin has activity toward cannabinoid receptor type 1 (CB1) with an IC50 value of 8.92 µM.	price>
R-C-2422	Varenicline Hydrochloride CAS:230615-23-3	Varenicline Hydrochloride(CP 526555 hydrochloride)is a high affinity, selective α4β2 nicotine acetylcholine receptor(nAChR)partial agonist and full α7 nAChR agonist.Varenicline Hydrochloride is also a potent partial agonist of α6β2 nAChR in striatum of rats with a Ki value of 0.12nM.	price>
R-R-4122	Arvanil CAS No.128007-31-8	Arvanil/CAS No.128007-31-8 is a ligand for vanilloid receptor 1 (VR1) and cannabinoid 1 (CB1). Arvanil can inhibit spasticity, as a potent neuroprotectant.	price>
R-C-2423	Myosmine CAS:532-12-7	Myosmine is not only one of the minor tobacco alkaloids but is also present in various foods.Myosmine has low affinity against a4b2 nicotinic acetylcholinergic receptors(nAChR)with Ki of 3300nM.	price>
R-R-4123	Taranabant ((1R,2R)stereoisomer) CAS No.701977-08-4	Taranabant (1R,2R)stereoisomer/CAS No.701977-08-4 is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist.	price>
R-C-2424	Amfebutamone (Bupropion) HCl CAS:31677-93-7	Amfebutamone(Bupropion)HCl is a selective norepinephrine-dopamine reuptake inhibitor with IC50 of 6.5 and 3.4uM for the reuptake of dopamine and norepinephrine,respectively.	price>
R-R-4124	Drinabant CAS No.358970-97-5	Drinabant (AVE1625)/CAS No.358970-97-5 is an orally active CB1 receptor antagonist. Drinabant (AVE1625) inhibits the agonist-stimulated calcium signal with IC50 values of 25 nM and 10 nM for the hCB1-R and rCB1-R, respectively, and is ineffective for the hCB2-R.	price>
R-C-2425	Galanthamine HBr CAS:1953-04-4	Galantamine Hydrobromide is the hydrobromide salt form of galantamine,a tertiary alkaloid with anticholinesterase and neurocognitive-enhancing activities.It is an alkaloid acetylcholinesterase inhibitor.Galantamine competitively and reversibly inhibits acetylcholinesterase,thereby increasing the concentration and enhancing the action of acetylcholine(Ach).	price>
R-R-4125	CB65 CAS No.913534-05-1	CB65/CAS No.913534-05-1 is a potent and high affinity CB2 selective agonist with a Ki value of 3.3 nM. CB65 exhibits a Ki of >1000 nM for CB1 receptor.	price>
R-C-2426	Rocuronium Bromide CAS:119302-91-9	Rocuronium Bromide is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia to facilitate endotracheal intubation by providing skeletal muscle relaxation.It is used for both standard and rapid sequence induction(RSI).	price>
R-R-4126	CB2R/FAAH modulator-3 CAS No.2876918-67-9	CB2R/FAAH modulator-3 (compound 27)/CAS No.2876918-67-9 is a dual targeting modulator that acts as a CB2R agonist and FAAH inhibitor. The Ki values for CB2R/FAAH modulator-3 are 20.1 and 67.6 nM for CB2R and CB1R, respectively, and the IC50 value for FAAH is 3.4 μM. CB2R/FAAH modulator-3 can be used in studies related to cancer, deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection.	price>
R-C-2427	Aclidinium Bromide CAS:320345-99-1	Aclidinium bromide is a long-acting anticholinergic bronchodilator approved by the FDA in 2012 for use in the management of chronic obstructive pulmonary disease(COPD)which includes chronic bronchitis and emphysema.	price>
R-R-4127	PGN36 CAS No.1564253-75-3	PGN36 (Compound 18)/CAS No.1564253-75-3 is a selective cannabinoid CB2 receptor (CB2R) antagonist with a Ki of 0.09 µM.	price>
R-C-2428	Otilonium Bromide CAS:26095-59-0	Otilonium bromide is an antimuscarinic and calcium channel blocker used to relieve spasmodic pain of the gut, especially in irritable bowel syndrome.	price>
R-R-4128	AM6545 CAS No.1245626-05-4	AM6545/CAS No.1245626-05-4 is a peripherally active, cannabinoid receptor antagonist with limited brain penetration. AM6545 binds to CB1 and CB2 receptors with Kis of 1.7 nM and 523 nM, respectively. AM6545 is a neutral antagonist. AM6545 can be used for the research of obesity and its complications.	price>
R-C-2429	Gallamine Triethiodide CAS:65-29-2	Gallamine Triethiodide is a mAChR M2 antagonist with pronounced cardioselectivity.It acts by combining with the cholinergic receptor sites in muscle and competitively blocks the transmitter action of acetylcholine.It is a synthetic non-depolarizing blocking drug.	price>
R-R-4129	2-Palmitoylglycerol CAS No.23470-00-0	2-Palmitoylglycerol (2-Palm-Gl)/CAS No.23470-00-0, an congener of 2-arachidonoylglycerol (2-AG), is a modest cannabinoid receptor CB1 agonist. 2-Palmitoylglycerol also may be an endogenous ligand for GPR119.	price>

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