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Catalog	name	Description	price
R-C-2416	Mirabegron CAS： 223673-61-8	Mirabegron(formerly YM-178,trade name Myrbetriq)is a drug for the treatment of overactive bladder.Mirabegron activates the β3 adrenergic receptor in the detrusor muscle in the bladder,which leads to muscle relaxation and an increase in bladder capacity.	price>
R-R-4116	2-Arachidonoylglycerol-d5 CAS No.2522598-88-3	2-Arachidonoylglycerol-d5/CAS No.2522598-88-3 is the deuterium labeled 2-Arachidonoylglycerol. 2-Arachidonoylglycerol is a second endogenous cannabinoid ligand in the central nervous system.	price>
R-C-2417	Olodaterol (BI 1744) CAS:868049-49-4	Olodaterol(BI 1744)is a long-acting β2-adrenergic receptor agonist that is used as a component of an inhalation(Tiotropium/Olodaterol)for treating patients with chronic obstructive pulmonary disease(COPD).	price>
R-R-4117	JTE-907 CAS No.282089-49-0	JTE-907/CAS No.282089-49-0 is a highly selective, orally active CB2 receptor inverse agonist and exerts anti-inflammatory effects in vivo.	price>
R-C-2418	Guanabenz CAS:5051-62-7	Guanabenz(Acetate)(BR-750)is an alpha-2 selective adrenergic agonist used as an antihypertensive agent.	price>
R-R-4118	GP1a CAS No.511532-96-0	GP1a/CAS No.511532-96-0 is a potent agonist of cannabinoid receptor 2 (CB2). Gp1a is beneficial to skin wound healing. GP1a inhibits inflammation and fibrogenesis while promoting re-epithelialization.	price>
R-C-2419	Droxidopa CAS:23651-95-8	Droxidopa is a synthetic amino acid precursor which acts as a prodrug to the neurotransmitters norepinephrine(noradrenaline)and epinephrine(adrenaline)and it is used to increase the concentrations of these neurotransmitters in the body and brain.Unlike norepinephrine and epinephrine themselves,droxidopa is capable of crossing the protective bloodÂ–brain barrier(BBB).	price>
R-R-4119	RVD-Hpα TFA CAS No.1431329-51-9	RVD-Hpα TFA/CAS No.1431329-51-9 is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. RVD-Hpα TFA increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. RVD-Hpα TFA also high affinity CB2 positive allosteric modulator (Ki=50 nM).	price>
R-C-2420	Dexmedetomidine CAS:113775-47-6	Dexmedetomidine is notable for its ability to provide sedation without risk of respiratory depression(unlike other commonly used sedatives such as propofol, fentanyl,and midazolam)and can provide cooperative or semi-arousable sedation.	price>
R-R-4120	BML-190 CAS No.2854-32-2	BML-190(IMMA)/CAS No.2854-32-2 is a potent and selective CB2 receptor ligand (Ki values are 435 nM and > 2 μM for CB2 and CB1 respectively).	price>
R-C-2421	Pimethixene maleate CAS:13187-06-9	Pimethixene(Pimetixene)maleate,an antihistamine,anntimigraine agent and antiserotonergic compound,is a highly potent antagonist of a broad range of monoamine receptors,including a variety of serotonin receptors.	price>
R-R-4121	Auriculasin CAS No.60297-37-2	Auriculasin/CAS No.60297-37-2 is a nature product isolated from Limonium leptophyllum. Auriculasin has activity toward cannabinoid receptor type 1 (CB1) with an IC50 value of 8.92 µM.	price>
R-C-2422	Varenicline Hydrochloride CAS:230615-23-3	Varenicline Hydrochloride(CP 526555 hydrochloride)is a high affinity, selective α4β2 nicotine acetylcholine receptor(nAChR)partial agonist and full α7 nAChR agonist.Varenicline Hydrochloride is also a potent partial agonist of α6β2 nAChR in striatum of rats with a Ki value of 0.12nM.	price>
R-R-4122	Arvanil CAS No.128007-31-8	Arvanil/CAS No.128007-31-8 is a ligand for vanilloid receptor 1 (VR1) and cannabinoid 1 (CB1). Arvanil can inhibit spasticity, as a potent neuroprotectant.	price>
R-C-2423	Myosmine CAS:532-12-7	Myosmine is not only one of the minor tobacco alkaloids but is also present in various foods.Myosmine has low affinity against a4b2 nicotinic acetylcholinergic receptors(nAChR)with Ki of 3300nM.	price>
R-R-4123	Taranabant ((1R,2R)stereoisomer) CAS No.701977-08-4	Taranabant (1R,2R)stereoisomer/CAS No.701977-08-4 is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist.	price>
R-C-2424	Amfebutamone (Bupropion) HCl CAS:31677-93-7	Amfebutamone(Bupropion)HCl is a selective norepinephrine-dopamine reuptake inhibitor with IC50 of 6.5 and 3.4uM for the reuptake of dopamine and norepinephrine,respectively.	price>
R-R-4124	Drinabant CAS No.358970-97-5	Drinabant (AVE1625)/CAS No.358970-97-5 is an orally active CB1 receptor antagonist. Drinabant (AVE1625) inhibits the agonist-stimulated calcium signal with IC50 values of 25 nM and 10 nM for the hCB1-R and rCB1-R, respectively, and is ineffective for the hCB2-R.	price>
R-C-2425	Galanthamine HBr CAS:1953-04-4	Galantamine Hydrobromide is the hydrobromide salt form of galantamine,a tertiary alkaloid with anticholinesterase and neurocognitive-enhancing activities.It is an alkaloid acetylcholinesterase inhibitor.Galantamine competitively and reversibly inhibits acetylcholinesterase,thereby increasing the concentration and enhancing the action of acetylcholine(Ach).	price>
R-R-4125	CB65 CAS No.913534-05-1	CB65/CAS No.913534-05-1 is a potent and high affinity CB2 selective agonist with a Ki value of 3.3 nM. CB65 exhibits a Ki of >1000 nM for CB1 receptor.	price>

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