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Catalog	name	Description	price
R-C-2426	Rocuronium Bromide CAS:119302-91-9	Rocuronium Bromide is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia to facilitate endotracheal intubation by providing skeletal muscle relaxation.It is used for both standard and rapid sequence induction(RSI).	price>
R-R-4126	CB2R/FAAH modulator-3 CAS No.2876918-67-9	CB2R/FAAH modulator-3 (compound 27)/CAS No.2876918-67-9 is a dual targeting modulator that acts as a CB2R agonist and FAAH inhibitor. The Ki values for CB2R/FAAH modulator-3 are 20.1 and 67.6 nM for CB2R and CB1R, respectively, and the IC50 value for FAAH is 3.4 μM. CB2R/FAAH modulator-3 can be used in studies related to cancer, deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection.	price>
R-C-2427	Aclidinium Bromide CAS:320345-99-1	Aclidinium bromide is a long-acting anticholinergic bronchodilator approved by the FDA in 2012 for use in the management of chronic obstructive pulmonary disease(COPD)which includes chronic bronchitis and emphysema.	price>
R-R-4127	PGN36 CAS No.1564253-75-3	PGN36 (Compound 18)/CAS No.1564253-75-3 is a selective cannabinoid CB2 receptor (CB2R) antagonist with a Ki of 0.09 µM.	price>
R-C-2428	Otilonium Bromide CAS:26095-59-0	Otilonium bromide is an antimuscarinic and calcium channel blocker used to relieve spasmodic pain of the gut, especially in irritable bowel syndrome.	price>
R-R-4128	AM6545 CAS No.1245626-05-4	AM6545/CAS No.1245626-05-4 is a peripherally active, cannabinoid receptor antagonist with limited brain penetration. AM6545 binds to CB1 and CB2 receptors with Kis of 1.7 nM and 523 nM, respectively. AM6545 is a neutral antagonist. AM6545 can be used for the research of obesity and its complications.	price>
R-C-2429	Gallamine Triethiodide CAS:65-29-2	Gallamine Triethiodide is a mAChR M2 antagonist with pronounced cardioselectivity.It acts by combining with the cholinergic receptor sites in muscle and competitively blocks the transmitter action of acetylcholine.It is a synthetic non-depolarizing blocking drug.	price>
R-R-4129	2-Palmitoylglycerol CAS No.23470-00-0	2-Palmitoylglycerol (2-Palm-Gl)/CAS No.23470-00-0, an congener of 2-arachidonoylglycerol (2-AG), is a modest cannabinoid receptor CB1 agonist. 2-Palmitoylglycerol also may be an endogenous ligand for GPR119.	price>
R-C-2430	Pyridostigmine Bromide CAS:101-26-8	Pyridostigmine Bromide is a cholinesterase inhibitor with a slightly longer duration of action than neostigmine.It is used in the treatment of myasthenia gravis and to reverse the actions of muscle relaxants.Pyridostigmine bromide binds reversibly to acetylcholinesterase active sites in the peripheral nervous system,thereby preventing the breakdown of acetylcholine. This leads to an accumulation of acetylcholine at cholinergic synapses and facilitates transmission of impulses across the neuromuscular junction.	price>
R-R-4130	CB-25 CAS No.869376-63-6	CB-25/CAS No.869376-63-6 is a ligand of CB1 cannabinoid receptors, acting as a partial agonist. CB-25 enhances Forskolin (HY-15371)-induced cAMP formation in cancer cells but not hCB1-CHO cells.	price>
R-C-2431	Rivastigmine Tartrate CAS:129101-54-8	Rivastigmine,also known as ENA-713,is a carbamate-derived reversible cholinesterase inhibitor that is selective for the central nervous system and is used for the treatment of Dementia,Alzheimer is Disease and Parkinson is Disease.It acts by covalently modifying a serine residue in the active site by carbamoylation,as it stabilizes or reduces the rate of decline in certain cognitive functions.	price>
R-R-4131	β-Caryophyllene-d2 CAS No.2006272-96-2	β-Caryophyllene-d2/CAS No.2006272-96-2 is deuterium labeled β-Caryophyllene. β-Caryophyllene is a CB2 receptor agonist.	price>
R-C-2432	Neostigmine Bromide CAS:114-80-7	Neostigmine bromide is a reversible inhibitor of acetylcholinesterase.AChE (acetylcholinesterase)is a hydrolase that hydrolyzes the neurotransmitter acetylcholine at the neuromuscular junction and cholinergic synaspe.It terminates the signal transductions and plays a role in neuronal apoptosis.	price>
R-R-4132	CB1/2 agonist 1	CB1/2 agonist 1 is a potent and cross the blood-brain barrier CB1/2 agonist with EC50s of 56.15, 11.63 nM for CB1R and CB2R, respectively. CB1/2 agonist 1 reduces glutamate release and LPS-induced activation of microglial cells. CB1/2 agonist 1 shows anti-inflammatory and antinociceptive effects. CB1/2 agonist 1 has the potential for the research of multiple sclerosis.	price>
R-C-2433	Donepezil CAS:120014-06-4	Donepezil is a noncompetitive acetylcholineesterase inhibitor,which can readily cross the blood brain barrier and increase the concentration of cortical acetylcholine.It is known that Donepezil is a useful tool in the study of Alzheimer is disease.	price>
R-R-4133	2-Linoleoyl glycerol CAS No.3443-82-1	3-Linoleoyl glycerol (2-Monolinolein; 2-Monolinoleoylglycerol)/CAS No.3443-82-1 is a monoacylglycerol that is an antagonist and partial agonist at the type 1 cannabinoid CB1 receptor. The potency of 2-Linoleoyl glycerol can be enhanced by JZL195 (HY-15250), an inhibitor of FAAH and MAGL, and inhibited by the CB1 antagonist AM251 (HY-15443) and Cannabidiol. As a CB1 antagonist, 2-Linoleoyl glycerol does not enhance, but only attenuates, the activity of the CB1/CB2 receptor ligands cannabinoids (AEA) and 2-arachidonoylglycerol (2-AG).	price>
R-C-2434	Nodakenetin CAS:495-32-9	Nodakenetin(NANI),a plant-derived coumarin isolated from Angelica decursiva, inhibits α-glucosidase,PTP1B,rat lens aldose reductase(RLAR),AChE,BChE,and β-site amyloid precursor protein cleaving enzyme 1(BACE1).Nodakenetin alters the protein expression of Bax and Bcl-2,and prompts mitochondrial apoptosis.Nodakenetin exhibits anti-tumor activity.	price>
R-R-4134	PSNCBAM-1 CAS No.877202-74-9	PSNCBAM-1/CAS No.877202-74-9 is a selective CB1 receptor allosteric antagonist with an EC50 of 0.1 μM. PSNCBAM-1 can be used in the researches of obesity.	price>
R-C-2435	Hyoscyamine CAS:101-31-5	Hyoscyamine is a tropane alkaloid.It is a secondary metabolite found in certain plants of the Solanaceae family.It is the levorotary isomer of atropine and thus sometimes known as levo-atropine.Hyoscyamine is used to provide symptomatic relief to various gastrointestinal disorders including spasms,peptic ulcers, irritable bowel syndrome,pancreatitis,colic and cystitis.	price>
R-R-4135	RTICBM-189 CAS No.551909-15-0	RTICBM-189/CAS No.551909-15-0 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay. RTICBM-189 has pIC50s of 5.29 and 6.25 for hCB1 and mCB1, respectively. RTICBM-189 significantly and selectively attenuates the reinstatement of the addictive agent-seeking behavior in rats.	price>

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