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Catalog	name	Description	price
R-C-2436	Huperzine B CAS:103548-82-9	Huperzine B is a efficient inhibitor of human brain AChE,it can enhance ognitive and protect neuro.	price>
R-R-4136	ZCZ011 CAS No.1998197-39-9	ZCZ011/CAS No.1998197-39-9 is a potent and brain penetrant cannabinoid 1 (CB1) receptor positive allosteric modulator. ZCZ011 potentiates binding of CP55,940 to the CB1 receptor, enhances anandamide (AEA)-stimulated GTPγS binding in mouse brain membranes. ZCZ011 increases β-arrestin recruitment and ERK phosphorylation in hCB1 cells. ZCZ011 can be used for researching neuropathic and inflammatory pain.	price>
R-C-2437	Picfeltarraenin IB CAS:97230-46-1	Picfeltarraenin IB,a cucurbitacin glycoside isolated from Picriafel-terrae,is an inhibitor of acetylcholinesterase(AChE).Picfeltarraenin IB can be used for the treatment of herpes infections,cancer and inflammation.	price>
R-R-4137	AEF0117 CAS No.1610878-71-1	AEF0117/CAS No.1610878-71-1 is a signaling-specific inhibitor of the cannabinoid receptor 1 (CB1-SSi). AEF0117 plays an important role in Cannabis use disorder (CUD).	price>
R-C-2438	Imidafenacin CAS:170105-16-5	Imidafenacin(KRP-197,ONO-8025)is a urinary antispasmodic of the anticholinergic class.Imidafenacin(KRP-197;ONO-8025)is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM;less potent for M2 receptors(IC50=4.13nM).IC50 value:0.3nM(M3).	price>
R-R-4138	CB2 receptor agonist 2 CAS No.1314230-75-5	CB2 receptor agonist 2/CAS No.1314230-75-5 is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor with a Ki of 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2.	price>
R-C-2439	Edrophonium chloride CAS:116-38-1	Edrophonium Chloride,also known as Tensilon,is an acetylcholinesterase inhibitor used in cardiac arrhythmias and in the diagnosis of myasthenia gravis. Edrophonium Chloride has also been used as an antidote to curare principles.	price>
R-R-4139	PSB-SB-487 CAS No.1399049-81-0	PSB-SB-487/CAS No.1399049-81-0 is a potent GPR55 antagonist and CB2 agonist with an IC50 value of 0.113 µM for GPR55, and a Ki value of 0.292 µM for human CB2. PSB-SB-487 can be used for researching diabetes, Parkinson’s disease, neuropathic pain, and cancer.	price>
R-C-2440	Corydaline CAS:518-69-4	Corydaline is a bioactive alkaloid with various anti-acetylcholinesterase,anti-allergic,and anti-nociceptive activities found in the medicinal herb Corydalis Tubers.	price>
R-R-4140	CB2 receptor agonist 3 CAS No.919077-81-9	CB2 receptor agonist 3/CAS No.919077-81-9 is a robust and selective CB2 cannabinoid agonist with Kis of 7.6 and 900 nM for CB2 and CB1, respectively. CB2 receptor agonist 3 significantly increases P-ERK 1/2 expression in HL-60 cells.	price>
R-C-2441	Atracurium Besylate CAS:64228-81-5	Atracurium Besilate is a neuromuscular-blocking drug or skeletal muscle relaxant in the category of non-depolarizing neuromuscular-blocking drugs,used adjunctively in anesthesia to facilitate endotracheal intubation and to provide skeletal muscle relaxation during surgery or mechanical ventilation.	price>
R-R-4141	(Rac)-Zevaquenabant CAS No.1610420-28-4	(Rac)-Zevaquenabant ((Rac)-MRI-1867/CAS No.1610420-28-4, compound 6b) is a cannabinoid receptor type 1 (CB1R)/iNOS antagonist, with a Ki of 5.7 nM for CB1R. (Rac)-Zevaquenabant is potential for the research of liver fibrosis.	price>
R-C-2442	Nodakenin CAS:495-31-8	Nodakenin acts as an AChE inhibitor that inhibits AChE activity in a dosedependent manner with an IC50 value of 84.7uM.Nodakenin possesses neuroprotective,anti-allergic,antiaggregatory,antibacterial,and memory -enhancing effects.Nodakenin down-regulates the expression of the proinflammatory iNOS,COX-2,TNF-α,IL-6,and IL-1β genes in macrophages by interfering with the activation of TRAF6,thus preventing NF-κB activation.	price>
R-R-4142	N-Arachidonyldopamine CAS No.199875-69-9	N-Arachidonyldopamine/CAS No.199875-69-9 is a potent and selective endogenous CB1 receptor agonist with a Ki of 250 nM. N-Arachidonyldopamine is also a potent and selective TRPV1 agonist an with EC50 of ~ 50 nM.	price>
R-C-2443	Loganin CAS:18524-94-2	Loganin(Loganoside)is an iridoid glycoside first isolated from the seeds of Strychnos nux-vomica,a member of the Loganiaceae family.It is a non-competitive inhibitor of BACE1 with IC50 of 47.97μM an also inhibits AChE and BChE with IC50 values of 3.95μM and 33.02μM, respectively.	price>
R-R-4143	CB2R/FAAH modulator-2 CAS No.2876918-68-0	CB2R/FAAH modulator-2 (compound 26)/CAS No.2876918-68-0 is a dual targeting modulator that acts as a CB2R agonist and FAAH inhibitor. The Ki values for CB2R/FAAH modulator-2 are 10.8 and 152.9 nM for CB2R and CB1R, respectively, and the IC50 value for FAAH is 6.2 μM. CB2R/FAAH modulator-2 can be used in studies related to cancer, deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection.	price>
R-C-2444	Palmatine CAS:3486-67-7	Palmatine(Berbericinine,Burasaine),an isoquinoline alkaloid,has sedative,antidepressant,antioxidative,anti-ulcerative,antacid,anticancer,and anti-metastatic activities.	price>
R-R-4144	CB1R antagonist 1 CAS No.334668-69-8	CB1R Allosteric modulator 5/CAS No.334668-69-8, a selective cannabinoid-1 receptor (CB1R) inverse agonist with an IC50 value of 4.2 μM and EC50 value of ＞10 μM. CB1R Allosteric modulator 5 can be used for the research of metabolic and obesity.	price>
R-C-2445	Jatrorrhizine chloride CAS:6681-15-8	Jatrorrhizine Chloride is a AChE inhibitor found in Corydalis and Coptydis.It increases expression of p21 and p27 and induces cell cycle arrest in melanoma cells,suppresses amyloid-β-induced toxicity in neurons,inhibits growth of Plasmodium,Leishmania,and Trypanosoma,and increases gastric emptying rates.	price>
R-R-4145	BMS-646256 CAS No.464213-10-3	BMS-646256/Ibipinabant/SLV319/CAS No.464213-10-3 is a potent, selective and orally active antagonist of cannabinoid CB1 receptor, with a Ki of 7.8 nM. Ibipinabant shows more than 1000-fold selectivity for CB1 over CB2 (Ki=7943 nM). Ibipinabant can be used for the research of obesity and diabetic.	price>

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