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Catalog	name	Description	price
R-R-4231	CCK-B Receptor Antagonist 2 CAS No.155412-88-7	CCK-B Receptor Antagonist 2/CAS No.155412-88-7, compound 15b, is a potent and orally active Gastrin/CCK-B antagonist with an IC50 value of 0.43 nM. CCK-B Receptor Antagonist 2 also inhibits gastrin/CCK-A activity with an IC50 of 1.82 μM.	price>
R-C-2532	APD668 CAS：832714-46-2	APD668 is a potent,selective and orally active agonist of G-protein coupled receptor GPR119,with EC50s of 2.7nM and 33nM for hGPR119 and rGPR119, respectively.APD668 shows no significant inhibition of any of the five major CYP isoforms with the exception of CYP2C9(Ki=0.1μM).APD668 can be used for the research of steatohepatitis and diabetes.	price>
R-R-4232	L-365260 hemihydrate	L-365260 hemihydrate is an orally active and selective antagonist of non-peptide gastrin and brain cholecystokinin receptor (CCK-B), with Kis of 1.9 nM and 2.0 nM, respectively. L-365260 hemihydrate interacts in a stereoselective and competitive manner with guinea pig stomach gastrin and brain CCK receptors.	price>
R-C-2533	Canagliflozin (JNJ 28431754) CAS：842133-18-0	Canagliflozin(JNJ 28431754)is a selective SGLT2 inhibitor with IC50s of 2nM, 3.7nM,and 4.4nM for mSGLT2,rSGLT2,and hSGLT2 in CHOK cells,respectively.	price>
R-R-4233	(Rac)-Sograzepide CAS No.168161-71-5	(Rac)-Sograzepide/CAS No.168161-71-5 is an antagonist of cholecystokinin B (CCK-B) receptor, and has the potential of reducing the secretion of gastric acid.	price>
R-C-2534	AMG073 CAS：226256-56-0	Cinacalcet(AMG073,Sensipar,Cin)is an orally active,allosteric agonist of receptors for calcium(CaR)that increases the sensitivity of the CaR to Ca.	price>
R-R-4234	CCK antagonist 1 CAS No.742116-45-6	CCK antagonist 1 (compound 3d)/CAS No.742116-45-6 is a CCK antagonist with IC50s of 1.1 μM and 4 μM for CCK1 and CCK2, respectively. CCK antagonist 1 can be used for research of cancer and mental disease.	price>
R-C-2535	Ambrisentan（BSF208075，LU208075） CAS No. 177036-94-1	Ambrisentan(LU-208075,BSF-208075)is a highly selective antagonist of the endothelin-1 type A receptor,used in the treatment of pulmonary arterial hypertension(PAH).	price>
R-R-4235	AMG 487 CAS No.473719-41-4	AMG 487/CAS No.473719-41-4 is an orally active and selective antagonist of CXC chemokine receptor 3 (CXCR3) which inhibits the binding of CXCL10 and CXCL11 to CXCR3 with IC50s of 8.0 and 8.2 nM, respectively.	price>
R-C-2536	Canagliflozin hemihydrate CAS：928672-86-0	Canagliflozin hemihydrate(JNJ28431754 hemihydrate) is a selective SGLT2 inhibitor with IC50s of 2nM,3.7nM,and 4.4nM for mSGLT2, rSGLT2,and hSGLT2 in CHOK cells,respectively.	price>
R-R-4236	Reparixin CAS No.266359-83-5	Reparixin/CAS No.266359-83-5 is a non-competitive allosteric inhibitor of the chemokine receptors CXCR1 and CXCR2 activation with IC50s of 1 and 100 nM, respectively.	price>
R-C-2537	Ipragliflozin (ASP1941) CAS：761423-87-4	Ipragliflozin(ASP1941)is an orally active and selective SGLT2 inhibitor with IC50s of 7.38 and 1876nM,6.73 and 1166nM,5.64 and 1380nM for human SGLT2 and SGLT1,rat SGLT2 and SGLT1,mouse SGLT2 and SGLT1,respectively.Antidiabetic agent.	price>
R-R-4237	Plerixafor octahydrochloride CAS No.155148-31-5	Plerixafor octahydrochloride (AMD3100 octahydrochloride)/CAS No.155148-31-5 is a selective CXCR4 antagonist with an IC50 of 44 nM.	price>
R-C-2538	Tofogliflozin(CSG 452) CAS：1201913-82-7	Tofogliflozin(CSG-452)is a potent and highly specific sodium/glucose cotransporter 2(SGLT2)inhibitor with Ki values of 2.9,14.9,and 6.4nM for human, rat,and mouse SGLT2.	price>
R-R-4238	Navarixin CAS No.473727-83-2	Navarixin (SCH 527123)/CAS No.473727-83-2 is a CXCR1 and CXCR2 antagonist that is potent, allosteric, and orally active, with Kd values of 41 nM for cynomolgus CXCR1 and 0.20 nM, 0.20 nM, 0.08 nM for mouse, rat and cynomolgus monkey CXCR2, respectively.	price>
R-C-2539	Plerixafor（ AMD310） CAS：110078-46-1	Plerixafor(AMD 3100)is a selective CXCR4 antagonist with an IC50 of 44nM.Plerixafor,an immunostimulant and a hematopoietic stem cell(HSC)mobilizer, is an allosteric agonist of CXCR7.Plerixafor inhibits HIV-1 and HIV-2 replication with an EC50 of 1-10nM.	price>
R-R-4239	AZD-5069 CAS No.878385-84-3	AZD-5069/CAS No.878385-84-3 is a potent CXCR2 chemokine receptor antagonist, used for caner treatment.	price>
R-C-2540	Ki16198 CAS：355025-13-7	Ki16198 is a potent and orally active LPA receptor antagonist,the methyl ester of Ki16425(HY-13285).Ki16198 inhibits LPA1 and LPA3-induced inositol phosphate production with Ki values of 0.34μM and 0.93μM,respectively.Ki16198 is effective for pancreatic cancer tumorigenesis and metastasis in vivo.	price>
R-R-4240	Mavorixafor trihydrochloride CAS No.2309699-17-8	Mavorixafor trihydrochloride (AMD-070 trihydrochloride)/CAS No.2309699-17-8 is a potent, selective and orally available CXCR4 antagonist, with an IC50 value of 13 nM against CXCR4 125I-SDF binding, and also inhibits the replication of T-tropic HIV-1 (NL4.3 strain) in MT-4 cells and PBMCs with an IC50 of 1 and 9 nM, respectively.	price>
R-C-2541	Oxiracetam CAS：62613-82-5	Oxiracetam is a cyclic derivative of γ-aminobutyric acid(GABA)which has been commonly used as nootropic drug to treat cognitive impairments.	price>

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