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Catalog	name	Description	price
R-C-2654	Satraplatin CAS:129580-63-8	Satraplatin(JM216,BMS182751)is a platinum compound that is currently under investigation as one treatment of patients with advanced prostate cancer who have failed previous chemotherapy.It has not yet received approval from the U.S.Food and Drug Administration.First mentioned in the medical literature in 1993,satraplatin is the first orally active platinum-based chemotherapeutic drug;other available platinum analogues-cisplatin,carboplatin,and oxaliplatin-must be given intravenously.	price>
R-R-4354	Molindone hydrochloride CAS No.15622-65-8	Molindone hydrochloride (EN-1733A)/CAS No.15622-65-8 is a therapeutic antipsychotic, used in the treatment of schizophrenia, works by blocking the effects of dopamine in the brain, leading to diminished psychoses.	price>
R-C-2655	INNO-206 CAS:1361644-26-9	Aldoxorubicin(INNO-206)is an albumin-binding prodrug of Doxorubicin(DNA topoisomerase II inhibitor),which is released from albumin under acidic conditions.Aldoxorubicin(INNO-206)has potent antitumor activities in various cancer cell lines and in murine tumor models.	price>
R-R-4355	ABT-724 trihydrochloride CAS No.587870-77-7	ABT-724 trihydrochloride/CAS No.587870-77-7 is a potent and highly selective dopamine D4 receptor agonist with an EC50 of 12.4 nM for human dopamine D4 receptor. ABT-724 trihydrochloride is a potent partial agonist at the rat D4 (EC50 of 14.3 nM) and the ferret D4 receptor (EC50 of 23.2 nM), and has no effect on dopamine D1, D2, D3, or D5 receptors. ABT-724 trihydrochloride could be useful for the treatment of erectile dysfunction and has favorable side-effect profile.	price>
R-C-2656	NVP-TNKS656 CAS:1419949-20-4	NVP-TNKS656 is a highly potent,selective,and orally active TNKS2 inhibitor with IC50 of 6nM,and is>300 fold selectivity against PARP1 and PARP2.	price>
R-R-4356	Bacopaside X CAS No.94443-88-6	Bacopaside X/CAS No.94443-88-6 is found in Bacopa monnieri, and shows a binding affinity toward the D1 receptor.	price>
R-C-2657	Dp44mT CAS: 152095-12-0	Dp44mT is an iron chelator,possessing DNA-damaging activity mediated by top2a inhibition.	price>
R-R-4357	Naxagolide CAS No.88058-88-2	Naxagolide ((+)-PHNO; Dopazinol)/CAS No.88058-88-2 is a potent dopamine D2 (Dopamine Receptor) agonist. Naxagolide has the potential for the research of parkinson disease (PD).	price>
R-C-2658	SCH 51344 CAS:171927-40-5	SCH-51344 is an inhibitor of RAS/RAC-mediated cell morphology pathway.RAS interacts with multiple targets in the cell and controls at least two signaling pathways,one regulating extracellular signal-regulated kinase(ERK)activation and the other controlling membrane ruffling formation.	price>
R-R-4358	JNJ-37822681 dihydrochloride CAS No.2108806-02-4	JNJ-37822681 dihydrochloride/CAS No.2108806-02-4 is a potent, specific, centrally active, fast-dissociating dopamine D2 receptor antagonist with a moderate binding affinity for the dopamine D2L receptor (Ki =158 nM), which has potential for the treatment of schizophrenia and bipolar disorder.	price>
R-C-2659	Apicidin CAS:183506-66-3	Apicidin(OSI 2040)is a fungal metabolite, acts as a histone deacetylase(HDAC)inhibitor,with antiparasitic activity and a broad spectrum antiproliferative activity.	price>
R-R-4359	(Rac)-Razpipadon CAS No.1643462-93-4	PW0464/CAS No.1643462-93-4, a nanomolar potent complete G protein biased ligand, is a noncatechol D1R agonist, with an EC50 of 5.8 nM (Gs-cAMP).	price>
R-C-2660	Triapine CAS：200933-27-3	Triapine(3-AP)is a potent ribonucleotide reductase(RNR)inhibitor with broad spectrum antitumor activity by inhibiting DNA synthesis.	price>
R-R-4360	MIF-1 TFA CAS No.35240-69-8	MIF-1 TFA (Melanostatin)/CAS No.35240-69-8, an endogenous brain peptide, is a potent dopamine receptor allosteric modulator. MIF-1 TFA inhibits melanin formation. MIF-1 TFA blocks the effects of opioid receptor activation to modulate the analgesic effects. MIF-1 TFA accesses from the blood to the CNS by directly crossing the blood-brain barrier (BBB).	price>
R-C-2661	Tasquinimod CAS：254964-60-8	Tasquinimod is an oral antiangiogenic agent,which has the potential for castration-resistant prostate cancer treatment.Tasquinimod binds to the regulatory Zn2+ binding domain of HDAC4 with Kd of 10-30nM.Tasquinimod also is a S100A9 inhibitor.	price>
R-R-4361	Alizapride hydrochloride CAS No.59338-87-3	Alizapride/CAS No.59338-87-3 is a potent antiemetic, acting as a dopamine receptor antagonist. Alizapride also used in human digestive disorders.	price>
R-C-2662	Paradol CAS:27113-22-0	Paradol is a pungent phenolic substance found in ginger and other Zingiberaceae plants.Paradol is an effective inhibitor of tumor promotion in mouse skin carcinogenesis,binds to cyclooxygenase(COX)-2 active site.	price>
R-R-4362	Aramisulpride CAS No.71675-90-6	Aramisulpride/CAS No.71675-90-6 is a dopamine D2 receptor and serotonin receptor antagonist used for the research of metabolic disorders.	price>
R-C-2663	XAV-939 CAS:284028-89-3	XAV-939 is a potent tankyrase inhibitor that targets Wnt/β-catenin signaling.XAV-939 stabilizes axin by inhibiting tankyrase 1 and tankyrase 2(IC50s of 5 and 2nM,respectively),thereby stimulating β-catenin degradation.XAV939 binds tightly to the catalytic(PARP)domains of TNKS1 and TNKS2(Kds of 99 and 93nM,respectively).	price>
R-R-4363	(R)-Preclamol hydrochloride CAS No.89874-80-6	(R)-Preclamol hydrochloride ((+)-3-PPP hydrochloride)/CAS No.89874-80-6 is the R-enantiomer of Preclamol hydrochloride. (R)-Preclamol hydrochloride is a DA agonist with autoreceptor as well as postsynaptic receptor stimulatory properties.	price>

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