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Catalog name Description price
R-C-2639 ZIP CAS:863987-12-6 ZIP is a selective peptide inhibitor of PKMζ.ZIP injections can block the impairment in morphine conditioned place preference induced. price>
R-R-4339 Tavapadon CAS No.1643489-24-0 Tavapadon (PF-06649751)/CAS No.1643489-24-0 is an orally active and highly selective dopamine D1/D5 receptor partial agonist. price>
R-C-2640 PPY A CAS:875634-01-8 PPY A is a potent inhibitor of T315l mutant and wild-type Abl kinases(IC50 values are 9 and 20nM,respectively).Inhibits growth of cells transformed with either the Bcr-Abl T315l mutant or wild-type Bcr-Abl gene. price>
R-R-4340 Mesdopetam hemitartrate CAS No.2562346-14-7 Mesdopetam (IRL790) hemitartrate/CAS No.2562346-14-7 is a dopamine D3 receptor antagonist (Ki=90 nM; IC50=9.8 μM for human recombinant D3 receptor) with psychomotor stabilizing properties. Mesdopetam hemitartrate is used for the research of motor and psychiatric complications in Parkinson disease. price>
R-C-2641 Bryostatin 2 CAS:87745-28-6 Bryostatin 2 is a protein kinase C(PKC)activator. price>
R-R-4341 Dopamine D2 receptor antagonist-1 CAS No.1055411-77-2 Dopamine D2 receptor antagonist-1/CAS No.1055411-77-2 is a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R) with sub-mM affinity. price>
R-C-2642 A 83-01 CAS: 909910-43-6 A 83-01 is a potent inhibitor of TGF-β type I receptor ALK5 kinase,type I nodal receptor ALK4 and type I nodal receptor ALK7,with IC50s of 12nM,45nM and 7.5nM against the transcription induced by ALK5,ALK4 and ALK7,respectively. price>
R-R-4342 Propionylpromazine hydrochloride CAS No.7681-67-6 Propionylpromazine hydrochloride (Propiopromazine hydrochloride)/CAS No.7681-67-6, a dopamine receptor D2 (DRD2) antagonist, can be used in the research of Parkinson disease. price>
R-C-2643 SPK-601 CAS:1096687-52-3 SPK-601(LMV-601)is an inhibitor of the phosphatidylcholine-specific phospholipase C(PC-PLC).SPK-601 also can be used as an antimicrobial agent. price>
R-R-4343 Quinelorane dihydrochloride CAS No.97548-97-5 Quinelorane dihydrochloride (LY163502)/CAS No.97548-97-5 is a potent dopamine D3/D2 receptor agonist. Quinelorane has the potential for neurological and psychiatric disorders research. price>
R-C-2644 Z-DEVD-FMK CAS:210344-95-9 Z-DEVD-FMK(Caspase-3 Inhibitor)is a specific,irreversible Caspase-3 inhibitor,and also shows potent inhibition on caspase-6,caspase-7,caspase-8, and caspase-10. price>
R-R-4344 (Rac)-PF-06256142 CAS No.1609580-97-3 (Rac)-PF-06256142/CAS No.1609580-97-3 is the less effective enantiomer of PF-06256142 (HY-119943). (Rac)-PF-06256142 is an agonist of D1 receptor, with an EC50 of 107 nM. price>
R-C-2645 Z-IETD-FMK CAS:210344-98-2 Z-IETD-FMK(Z-IE(OMe)TD(OMe)-FMK)is a selective and cell permeable caspase-8 inhibitor.Z-IETD-FMK is also a granzyme B inhibitor. price>
R-R-4345 Carmoxirole hydrochloride CAS No.115092-85-8 Carmoxirole hydrochloride (EMD 45609 hydrochloride)/CAS No.115092-85-8 is a selective, peripherally acting dopamine D2 receptor agonist and exhibits antihypertensive activities in vivo. price>
R-C-2646 Z-WEHD-FMK CAS:210345-00-9 Z-WEHD-FMK is a potent,cell-permeable and irreversible caspase-1/5 inhibitor.Z-WEHD-FMK also exhibits a robust inhibitory effect on cathepsin B activity (IC50=6μM).Z-WEHD-FMK can be used to investigate cells for evidence of apoptosis. price>
R-R-4346 Acetophenazine dimaleate CAS No.5714-00-1 Acetophenazine dimaleate/CAS No.5714-00-1, a phenothiazine derivative, is an antipsychotic agent. Acetophenazine dimaleate primarily blocks dopamine D2 receptors in the brain. Acetophenazine dimaleate can be used for researching psychotic disorders such as schizophrenia and anxious depression. price>
R-C-2647 Ac-LEHD-AFC Ac-LEHD-AFC,fluorogenic caspase substrate.Analog of the caspase-9 substrate, LEHD-AFC. price>
R-R-4347 UCM-1306 CAS No.2258608-78-3 UCM-1306/CAS No.2258608-78-3 is a potent and orally active human dopamine D1 receptor allosteric modulator (PAM). UCM-1306 increases the endogenous dopamine (DA) maximal effect both in human and mouse D1 receptors. UCM-1306 is not only for improving motor symptoms but also for addressing the key comorbid cognitive impairment associated with long-term Parkinson disease (PD). price>
R-C-2648 Gambogic acid CAS:2752-65-0 Gambogic Acid(Beta-Guttiferrin)is derived from the gamboges resin of the tree Garcinia hanburyi.Gambogic Acid (Beta-Guttiferrin)inhibits Bcl-XL,Bcl-2,Bcl-W,Bcl-B,Bfl-1 and Mcl-1 with IC50s of 1.47μM,1.21μM,2.02 μM,0.66μM,1.06μM and 0.79μM. price>
R-R-4348 L-745870 hydrochloride CAS No.1173023-36-3 L-745870 hydrochloride/CAS No.1173023-36-3 is a potent, selective, brain-penetrant and orally active dopamine D4 receptor antagonist with a Ki of 0.43 nM. L-745870 hydrochloride shows weaker affinity for D2 (Ki of 960 nM) and D3 (Ki of 2300 nM) receptors, and exhibits moderate affinity for 5-HT2 receptors, sigma sites and α-adrenoceptors. price>