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Catalog	name	Description	price
R-R-4371	L-DOPA-d6 CAS No.713140-75-1	L-DOPA-d6/CAS No.713140-75-1 is the deuterium labeled L-DOPA. L-DOPA (Levodopa) is an orally active metabolic precursor of neurotransmitters dopamine. L-DOPA can cross the blood-brain barrier and is converted into dopamine in the brain.	price>
R-C-2672	Flumequine CAS:42835-25-6	Flumequine(R-802)is a quinolone antibiotic,and acts as a topoisomerase II inhibitor,with an IC50 of 15μM(3.92μg/mL).	price>
R-R-4372	Odapipam CAS No.131796-63-9	Odapipam (NNC 756)/CAS No.131796-63-9 is a selective, high affinity and benzazepine dopamine D1 receptor antagonist with a Kd of 0.18 nM. Odapipam is also a superior positron emission tomography (PET) radiotracer.	price>
R-C-2673	Beta-Lapachone CAS:4707-32-8	Beta-Lapachone is a selective DNA topoisomerase I inhibitor,exhibiting no inhibitory activities against DNA topoisomerase II or ligase.	price>
R-R-4373	Preclamol hydrochloride CAS No.88768-67-6	Preclamol hydrochloride ((-)-3-PPP hydrochloride)/CAS No.88768-67-6 is a selective dopamine autoreceptor agonist. Preclamol hydrochloride has the potential for the research of schizophrenia.	price>
R-C-2674	Floxuridine CAS:50-91-9	Floxuridine(NSC 27640,Deoxyfluorouridine,FUDR)is a prodrug that is rapidly catabolized to 5-fluorouracil in vivo.Floxuridine inhibits Poly(ADP-Ribose) polymerase and induces DNA damage and apoptosis.Floxuridine has antiviral effects against HSV and CMV.	price>
R-R-4374	Etilevodopa hydrochloride CAS No.39740-30-2	Etilevodopa (L-Dopa ethyl ester) hydrochloride/CAS No.39740-30-2, an ethyl-ester proagent of Levodopa, is rapidly hydrolyzed to Levodopa and ethanol by nonspecific esterases in the gastrointestinal tract. Etilevodopa hydrochloride is used for the treatment of Parkinson disease (PD). Levodopa is the direct precursor of dopamine and is a suitable proagent as it facilitates CNS penetration and delivers dopamine.	price>
R-C-2675	Ellipticine CAS：519-23-3	Ellipticine is a DNA intercalating agent and a DNA topoisomerase II inhibitor.	price>
R-R-4375	GBR 12783 dihydrochloride CAS No.67469-75-4	GBR 12783 dihydrochloride/CAS No.67469-75-4 is a specific, potent and selective dopamine uptake inhibitor that inhibits the [3H]dopamine uptake by rat and mice striatal synaptosomes with IC50s of 1.8 nM and 1.2 nM, respectively. GBR 12783 dihydrochloride can improve memory performance and increase hippocampal acetylcholine release in rats.	price>
R-C-2676	Costunolide CAS：553-21-9	Costunolide(NSC 106404),a natural sesquiterpene compound with multiple biological activities;inhibits FPTase with IC50 of 20μM,also inhibits telomerase with IC50 of 65-90μM.	price>
R-R-4376	Veralipride CAS No.66644-81-3	Veralipride/CAS No.66644-81-3 is a D2 receptor antagonist. It is an alternative antidopaminergic treatment for menopausal symptoms.	price>
R-C-2677	KU 55933 CAS：587871-26-9	KU-55933 is an ATM inhibitor,which blocks the phosphorylation of Akt induced by insulin and insulin-like growth factor I in cancer cells that exhibit abnormal Akt activity. Moreover,KU-55933 inhibits cancer cell proliferation by inducing G(1)cell cycle arrest.It does so through the downregulation of the synthesis of cyclin D1,a protein known to be elevated in a variety of tumors.	price>
R-R-4377	(R)-Preclamol CAS No.85976-54-1	(R)-Preclamol/CAS No.85976-54-1 is a dopamine (DA) agonist with autoreceptor as well as postsynaptic receptor stimulatory properties. (R)-Preclamol inhibits the locomotor activity of mice and rats in low doses.	price>
R-C-2678	Trichostatin A (TSA) CAS：58880-19-6	Trichostatin A(TSA)is a potent and specific inhibitor of HDAC class I/II,with an IC50 value of 1.8nM for HDAC.	price>
R-R-4378	SKF-75670 hydrobromide CAS No.62717-63-9	SKF-75670 hydrochloride/CAS No.62717-63-9 is a Dopamine D1 receptor partial agonist. SKF-75670 hydrochloride is also a Cocaine antagonist.	price>
R-C-2679	Carmofur CAS：61422-45-5	Carmofur(HCFU),a derivative of 5-Fluorouracil,is an antineoplastic agent.Carmofur is an inhibitor of acid ceramidase with an IC50 of 79nM for the rat enzyme.Carmofur inhibits the SARS-CoV-2 main protease(Mpro).Carmofur Inhibits SARS-CoV-2 in Vero E6 cell with an EC50 of 24.3μM.	price>
R-R-4379	Bromopride CAS No.4093-35-0	Bromopride/CAS No.4093-35-0 is a dopamine antagonist with prokinetic properties, widely used as an antiemetic.	price>
R-C-2680	Altretamine CAS：645-05-6	Altretamine is classified as an alkylating antineoplastic agent.This unique structure is believed to damage tumor cells through the production of the weakly alkylating species formaldehyde,a product of CYP450-mediated N-demethylation.	price>
R-R-4380	Ziprasidone amino acid CAS No.1159977-64-6	Ziprasidone amino acid (Ziprasidone Impurity C)/CAS No.1159977-64-6 is an impurity of Ziprasidone. Ziprasidone is a combined 5-HT (serotonin) and dopamine receptor antagonist. Ziprasidone exhibits potent effects of antipsychotic activity .	price>
R-C-2681	Amonafide CAS： 69408-81-7	Amonafide is a topoisomerase II inhibitor and DNA intercalator that induces apoptotic signaling by blocking the binding of Topo II to DNA.	price>

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