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Catalog name Description price
R-R-3950 Midodrine-d6 hydrochloride CAS No.1188265-43-1 Midodrine-d6 (hydrochloride)/CAS No.1188265-43-1 is deuterium labeled Midodrine, which is a vasopressor/antihypotensive agent. price>
R-R-3951 Vilanterol-d4 trifenatate CAS No.2021249-10-3 Vilanterol-d4 (trifenatate)/CAS No.2021249-10-3 is deuterium labeled Vilanterol (trifenatate). Vilanterol trifenatate (GW642444 trifenatate) is a long-acting β2-adrenoceptor (β2-AR) agonist with inherent 24-hour activity. The pEC50s for β2-AR, β1-AR and β3-AR are 10.37, 6.98 and 7.36, respectively. price>
R-R-3952 Oxprenolol-d7 CAS No.1189805-10-4 Oxprenolol-d7/CAS No.1189805-10-4 is the deuterium labeled Oxprenolol. Oxprenolol (Ba 39089 free base) is an orally bioavailable β-adrenergic receptor (β-AR) antagonist with a Ki of 7.10 nM in a radioligand binding assay using rat heart muscle. price>
R-R-3953 Brimonidine-d4 CAS No.1184971-51-4 Brimonidine-d4/CAS No.1184971-51-4 is the deuterium labeled Brimonidine. Brimonidine (UK 14304) is a full α2-adrenergic receptor (α2-AR) agonist. price>
R-R-3954 Benoxathian hydrochloride CAS No.92642-97-2 Benoxathian hydrochloride/CAS No.92642-97-2 is a potent α1 adrenoceptor antagonist, can be used for researching anorexia. price>
R-R-3955 Brimonidine-d4 D-tartrate CAS No.1316758-27-6 Brimonidine-d4 (D-tartrate)/CAS No.1316758-27-6 is the deuterium labeled Brimonidine D-tartrate. price>
R-R-3956 Tetrahydrozoline-d4 hydrochloride CAS No.1246814-66-3 Tetrahydrozoline-d4 (hydrochloride)/CAS No.1246814-66-3 is the deuterium labeled Tetrahydrozoline hydrochloride. Tetrahydrozoline hydrochloride (Tetryzoline hydrochloride), a derivative of imidazoline, is an α-adrenergic agonist that causes vasoconstriction. Tetrahydrozoline hydrochloride is widely used for the research of nasal congestion and conjunctival congestion. price>
R-R-3957 ST91 CAS No.4749-61-5 ST91/CAS No.4749-61-5 is a α2-adrenoceptor (α2AR) agonist. ST91 activates both α2AAR and non-α2AAR subtypes to produce spinal antinociception. price>
R-R-3958 Octopamine-d4 hydrochloride CAS No.1219803-62-9 Octopamine-d4 (hydrochloride)/CAS No.1219803-62-9 is the deuterium labeled Octopamine hydrochloride. Octopamine ((±)-p-Octopamine) hydrochloride, a biogenic monoamine structurally related to noradrenaline, acts as a neurohormone, a neuromodulator and a neurotransmitter in invertebrates. Octopamine hydrochloride can stimulate alpha2-adrenoceptors (ARs) in Chinese hamster ovary cells transfected with human alpha2-ARs. Octopamine hydrochloride increased glycogenolysis, glycolysis, oxygen uptake, gluconeogenesis and the portal perfusion pressure. price>
R-R-3959 Amitriptyline hydrochloride (Standard) CAS No.549-18-8 Amitriptyline (hydrochloride) (Standard)/CAS No.549-18-8 is the analytical standard of Amitriptyline (hydrochloride). This product is intended for research and analytical applications. Amitriptyline hydrochloride is an inhibitor of serotonin reuptake transporter (SERT) and noradrenaline reuptake transporter (NET), with Kis of 3.45 nM and 13.3 nM for human SERT and NET, respectively. Amitriptyline hydrochloride also weakly binds to dopamine reuptake transporter (DAT) with a Ki of 2.58 μM. Amitriptyline hydrochloride also inhibits adrenergic, muscarinic, histamine and 5-HT receptors. Amitriptyline hydrochloride is a TrkA and TrkB receptors agonist with potent neurotrophic activity. Amitriptyline hydrochloride has antidepressant activity. price>