Product apis-gpcr-g-protein

Home > products > apis> gpcr-g-protein

Catalog	name	Description	price
R-R-3610	Vilanterol CAS No.503068-34-6	Vilanterol (GW642444)/CAS No.503068-34-6 is a long-acting β2-adrenoceptor (β2-AR) agonist with 24 h activity. The pEC50s for β2-AR,β1-AR and β3-AR is 10.37±0.05, 6.98±0.03 and 7.36±0.03, respectively.	price>
R-R-3611	(R)-Propranolol hydrochloride CAS No.13071-11-9	(R)-Propranolol hydrochloride/CAS No.13071-11-9 is a less active enantiomer of the β-adrenoceptor antagonist propranolol (HY-B0573). Propranolol is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively.	price>
R-R-3612	Rauwolscine hydrochloride CAS No.6211-32-1	Rauwolscine hydrochloride/CAS No.6211-32-1 is a potent and specific α2 adrenergic receptor antagonist with a Ki of 12 nM.	price>
R-R-3613	Acebutolol hydrochloride CAS No.34381-68-5	Acebutolol hydrochloride/CAS No.34381-68-5 is an orally active β1 adrenergic receptor (β1AR) antagonist. Acebutolol hydrochloride is used in the treatment of hypertension, angina pectoris and cardiac arrhythmias.	price>
R-C-1914	LY2795050 CAS：1346133-08-1	LY2795050 is a novel selective κ-opioid Receptor(KOR)antagonist(IC50=0.72nM) and has the potential as a PET tracer to image KOR in vivo.	price>
R-R-3614	Midodrine hydrochloride CAS No.43218-56-0	Midodrine hydrochloride ((±)-Midodrine hydrochloride)/CAS No.43218-56-0 is an α1-receptor agonist, for the treatment of dysautonomia and orthostatic hypotension.	price>
R-R-3615	Penbutolol sulfate CAS No.38363-32-5	Penbutolol sulfate/CAS No.38363-32-5 is able to bind to both beta-1 adrenergic receptors and beta-2 adrenergic receptors (the two subtypes), thus making it a non-selective β blocker.	price>
R-R-3616	JP1302 dihydrochloride CAS No.1259314-65-2	JP1302 dihydrochloride/CAS No.1259314-65-2 is a potent, selective, high affinity antagonist of the α2C-adrenoceptor, with a Kb of 16 nM and a Ki of 28 nM for the human α2C-receptor. JP1302 dihydrochloride shows antidepressant and antipsychotic-like effects. JP1302 dihydrochloride can be used for neuropsychiatric disorders and renal dysfunction research.	price>
R-R-3617	Medetomidine hydrochloride CAS No.86347-15-1	Medetomidine hydrochloride/CAS No.86347-15-1 is an orally active α2-adrenoceptor agonist (Ki: 1.08 nM). Medetomidine hydrochloride has sedative and analgesic effects. Medetomidine hydrochloride can cause peripheral vasoconstriction through the activation of α2 adrenoceptors on blood vessels.	price>
R-R-3618	2-Methoxyidazoxan monohydrochloride CAS No.109544-45-8	2-Methoxyidazoxan monohydrochloride (RX821002 hydrochloride)/CAS No.109544-45-8 is a highly selective alpha 2-adrenoceptor antagonist with little or no imidazoline antagonist effect. RX 821002 has markedly higher affinity for (guinea-pig) alpha 2D-adrenoceptors (pKd 9.7) than for (rabbit) alpha 2A-adrenoceptors (pKd 8.2).	price>

...

163