Product apis-ubiquitin

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Catalog	name	Description	price
R-C-3104	PYR-41 CAS:418805-02-4	PYR-41 is the first cell-permeable inhibitor of ubiquitin-activating enzyme E1, with no activity at E2.PYR-41 induce apoptosis.	price>
R-C-3105	BAY 11-7082 (BAY 11-7821) CAS:19542-67-7	BAY 11-7082(BAY 11-7821)is a NF-κB inhibitor, inhibits TNFα-induced IκBα phosphorylation with IC50 of 10μM in tumor cells. BAY 11-7082 inhibits ubiquitin-specific protease USP7 and USP21 with IC50 of 0.19 μM and 0.96 μM,respectively.BAY 11-7082 induces apoptosis and S phase arrest in gastric cancer cells.	price>
R-C-3106	TZ9 CAS:1002789-86-7	TZ9 is a novel inhibitor of Rad6 ubiquitin conjugating enzyme(E2 enzyme); inhibits MDA-MB-231 cell proliferation with IC50 of ~6 uM.	price>
R-C-3107	HLI-98C CAS:317326-90-2	HLI-98C,an analog,indeed inhibited Mdm2 E3 ligase activity.	price>
R-C-3108	TAME CAS:901-47-3	TAME is a small molecule anaphase-promoting complex/cyclosome(APC)inhibitor with an IC50 of 12μM.	price>
R-C-3109	SMER3 CAS:67200-34-4	SMER3 is a selective inhibitor of a yeast SCF family E3 ubiquitin ligase(SCFMet30)in vitro and in vivo. Induces the expression of MET genes;blocks cell proliferation.	price>
R-C-3111	SJB3-019A CAS: 2070015-29-9	SJB3-019A,also known as SJB 019, is a USP1 inhibitor.	price>
R-C-3112	DUBs-IN-1 CAS:924296-18-4	DUBs-IN-1 is a potent deubiquitinase enzyme inhibitor with IC50s of 18 uM/0.71 uM for USP7/USP8 respectively.	price>
R-C-3113	DUBs-IN-3 CAS：924296-17-3	DUBs-IN-3 is a potent deubiquitinase enzyme inhibitor with IC50s of 3.1uM for USP8;>30 fold selectivity over USP7 (IC50>100uM).	price>
R-C-3114	GNE-6640 CAS：2009273-67-8	GNE-6640 is a selective and non-covalent inhibitor of ubiquitin epecific peptidase 7 (USP7), with IC50 values of 0.75 μM,0.43 μM,20.3μM and 0.23μM for full length USP7, USP7 catalytic domain, full length USP43 and Ub-MDM2,respectively.	price>

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