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GSK973 CAS No.2138473-38-6

Catalog #	Pkg Size	Price(USD)	Quantity	Buy this product
R-R-2595	5mg	340.00	- +	+ Add to cart
R-R-2595	10mg	580.00	- +	+ Add to cart

Product description

GSK973/CAS No.2138473-38-6 is a highly selective, orally bioavailable inhibitor of the BD2s (second bromodomains) of the BET family, with a pIC50 of 7.8 and a pKd of 8.7 for BRD4 BD2. GSK973 displays a 1600-fold selectivity for BRD4 BD2 over BRD4 BD1. GSK973 shows good potency against BRD2 BD2, BRD3 BD2, and BRDT BD2 (pIC50=7.4~7.8; pKd=8.3~8.5).

Appearance	N/A
Molecular Weight	410.44
Purity	>90%
CAS	2138473-38-6
Formula	C23H23FN2O4
Storage	-20℃, protected from light and moisture
Transportation	4-25℃ temperature for up to 2 weeks
Stability	1 year

Document

msds of GSK973 CAS No.2138473-38-6