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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-3788 Metipranolol CAS No.22664-55-7 Metipranolol/CAS No.22664-55-7 is a nonselective and orally active β-adrenergic receptor antagonist. Metipranolol can be used for hypertension and glaucoma research. price>
R-R-3789 Denopamine CAS No.71771-90-9 Denopamine ((R)-(-)-Denopamine)/CAS No.71771-90-9 is an orally active, selective β1-adrenergic agonist. Denopamine prolongs survival in a murine model of congestive heart failure induced by viral myocarditis: suppression of tumor necrosis factor-α production in the heart. Cardiovascular effects. price>
R-R-3790 DL-Norepinephrine-d6 hydrochloride CAS No.1219803-04-9 DL-Norepinephrine-d6 (hydrochloride)/CAS No.1219803-04-9 is the deuterium labeled DL-Norepinephrine hydrochloride. DL-Norepinephrine hydrochloride is a synthetic phenylethylamine that mimics the sympathomimetic actions of the endogenous norepinephrine．DL-Norepinephrine hydrochloride is a neurotransmitter targets α1 and β1 adrenoceptors, has an increasing effect on subendocardial oxygen tension. price>
R-R-3791 Atenolol-d7 CAS No.1202864-50-3 Atenolol-d7/CAS No.1202864-50-3 is the deuterium labeled Atenolol. Atenolol ((RS)-Atenolol) is a cardioselective β1-adrenergic receptor blocker, with a Ki of 697 nM atβ1-adrenoceptor in guine pig left ventricle membrane. Atenolol can be used for the research of hypertension and angina pectoris. price>
R-R-3792 Bretylium tosylate CAS No.61-75-6 Bretylium (tosylate)/CAS No.61-75-6 is an inhibitor of the presynaptic release of vasoconstrictor neurotransmitters. price>
R-R-3793 Etilefrine hydrochloride CAS No.943-17-9 Etilefrine hydrochloride/CAS No.943-17-9 is an orally active α adrenergic agonist. Etilefrine hydrochloride is also an AMPK activator. Etilefrine hydrochloride can be used for the research of postural hypotension. price>
R-R-3794 CGP 20712 A CAS No.105737-62-0 CGP 20712 A (CGP 20712 mesylate)/CAS No.105737-62-0 is a highly selective β1-adrenoceptor antagonist with an IC50 of 0.7 nM. CGP 20712 A exhibits ~10,000-fold selectivity over β2-adrenoceptors. price>
R-R-3795 ONO-2952 CAS No.895169-20-7 ONO-2952/CAS No.895169-20-7 is a potent, selective and orally active translocator protein 18 kDa (TSPO) antagonist with Ki of 0.33-9.30 nM for rat and human TSPO. ONO-2952 is more selective for TSPO than other receptors, transporters, ion channels and enzymes. ONO-2952 exerts its anti-stress effects through inhibition of excessive activation of noradrenergic system in the brain without the amnesic effect. ONO-2952 has the potential for irritable bowel syndrome treatment. price>
R-R-3796 Centanafadine hydrochloride CAS No.923981-14-0 Centanafadine (hydrochloride)/CAS No.923981-14-0 is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter , respectively. price>
R-R-3797 Vanilpyruvic acid CAS No.1081-71-6 Vanilpyruvic acid/CAS No.1081-71-6 is a catecholamine metabolite and precursor to vanillactic acid. price>