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Catalog name Description price
R-R-3798 Clorprenaline hydrochloride CAS No.6933-90-0 Clorprenaline hydrochloride/CAS No.6933-90-0 is a β2-adrenergic receptor agonist that is implicated in bronchial expansion. Clorprenaline has the potential for asthma research. price>
R-R-3799 Guanadrel CAS No.40580-59-4 Guanadrel/CAS No.40580-59-4 is an orally active postganglionic adrenergic inhibitor of spiroketal. Guanadre can be used in anti-hypertensive studies. price>
R-R-3800 LY377604 CAS No.204592-94-9 LY377604/CAS No.204592-94-9 is a human β3-adrenergic receptor agonist with an EC50 of 2.4 nM and also a β1- and β2-adrenergic receptor antagonist. price>
R-C-2101 BAY-545 CAS：1699717-32-2 BAY-545 is a potent and selective A2B adenosine receptor antagonist, with an IC50 of 59 nM. BAY-545 also exhibits IC50s of 66,400,280 nM for human, mouse,rat A2B adenosine receptor in cells,respectively,and a Ki of 97nM for human A2B adenosine receptor,with more selectivity over A1,A2A,and A3 adenosine receptor. price>
R-R-3801 Apraclonidine hydrochloride CAS No.73218-79-8 Apraclonidine hydrochloride (ALO 2145)/CAS No.73218-79-8, a selective α2 and weak α1 receptor agonist activity, effectively lowers intraocular pressure (IOP) in human eyes. Apraclonidine hydrochloride is a topical ophthalmic solution and has the ability to elevate the eye lid. price>
R-R-3802 Tizanidine hydrochloride CAS No.64461-82-1 Tizanidine hydrochloride/CAS No.64461-82-1 is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons. price>
R-R-3803 Lofexidine hydrochloride CAS No.21498-08-8 Lofexidine (hydrochloride)/CAS No.21498-08-8 is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal. price>
R-C-2104 BAR 502 CAS：1612191-86-2 BAR502 is a dual FXR and GPBAR1 agonist.BAR-502 promotes browning of white adipose tissue and reverses liver steatosis and fibrosis.BAR502 protects against liver damage caused by HFD by promoting the browning of adipose tissue. price>
R-R-3804 Ritodrine hydrochloride CAS No.23239-51-2 Ritodrine (DU21220) hydrochloride/CAS No.23239-51-2 is a β-adrenergic agonist, also an effective smooth muscle and uterine relaxant. Ritodrine hydrochloride prolongs contraction interval, can be used for researching arrest premature labor. price>
R-C-2105 BAR 501 CAS： 1632118-69-4 BAR501 is a potent and selective G protein-coupled bile acid receptor 1(GPBAR1, GPCR19,TGR5)agonist that effectively transactivates GPBAR1 in HEK293 cells overexpressing a CRE along with GPBAR1 with EC50 of 1μM. price>