Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3401	MS 245 oxalate CAS No.275363-58-1	MS 245 oxalate/CAS No.275363-58-1 is a potent antagonist of 5-HT6 receptor with a Ki of 2 nM.	price>
R-R-3402	Blonanserin-d5 CAS No.1346599-86-7	Blonanserin-d5/CAS No.1346599-86-7 is a deuterium labeled Blonanserin. Blonanserin is a dopamine D2/5-HT2 receptor antagonist and an atypical antipsychotic.	price>
R-R-3403	SB-216641A CAS No.193611-67-5	SB-216641A (SB-216641 hydrochloride)/CAS No.193611-67-5 is a selective antagonist of 5-HT1B/D receptor. SB-216641A shows high affinity and selectivity for h5-HT1B receptors over h5-HT1D receptors. SB-216641A inhibits the function of SKF-99101H.	price>
R-R-3404	Cyproheptadine-d3 CAS No.2712455-05-3	Cyproheptadine-d3/CAS No.2712455-05-3 is deuterium labeled Cyproheptadine.	price>
R-R-3405	Robalzotan hydrochloride CAS No.184674-99-5	Robalzotan hydrochloride (NAD-299 hydrochloride)/CAS No.184674-99-5 is a potent and selective 5-Hydroxytryptamine 1A (5-HT1A) inhibitor. Robalzotan hydrochloride increases the firing rate of 5-HT cells. Robalzotan hydrochloride induces 5-HT1A receptor occupancy. Robalzotan hydrochloride has the potential for the research of a cholinergic deficit in the central -nervous system.	price>
R-R-3406	(Rac)-Rotigotine CAS No.92206-54-7	(Rac)-Rotigotine (N-0437)/CAS No.92206-54-7 is a racemate of Rotigotine. Rotigotine is a full agonist of?dopamine receptor, a partial agonist of the?5-HT1A receptor, and an antagonist of the?α2B-adrenergic receptor, with?Kis of 0.71?nM, 4-15?nM, and 83?nM for the dopamine D3 receptor and D2, D5, D4 receptors, and dopamine D1 receptor.	price>
R-R-3407	LY320135 CAS No.176977-56-3	LY320135/CAS No.176977-56-3 is a potent and selective antagonist of CB1 receptor, with a Ki of 141 nM. LY320135 also binds to 5-HT2 and muscarinic receptors with Kis of 6.4 μM and 2.1 μM, respectively. LY320135 exhibits neuroprotective effect.	price>
R-R-3408	U92016A hydrochloride CAS No.149654-41-1	U92016A hydrochloride/CAS No.149654-41-1 is a potent, metabolically stable, orally acitive 5-HT1A receptor agonist with an exceptionally high degree of intrinsic activity. U92016A hydrochloride binds with high affinity to human 5-HT1A receptors expressed in Chinese hamster ovary cells (Ki=0.2 nM).	price>
R-R-3409	PRX933 hydrochloride CAS No.639029-42-8	PRX933 hydrochloride/CAS No.639029-42-8 is a 5-HT2c receptor agonist extracted from patent WO 2014140631 A1.	price>
R-R-3410	Norfluoxetine-d5 hydrochloride CAS No.1188265-34-0	Norfluoxetine-d5 (hydrochloride)/CAS No.1188265-34-0 is deuterium labeled 3-Phenyl-3-(4-(trifluoromethyl)phenoxy)propan-1-amine hydrochloride.	price>

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