Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-3383	Ipsapirone CAS No.95847-70-4	Ipsapirone (TVX Q 7821)/CAS No.95847-70-4 is an anxiolytic compound and a 5-HT1A receptor partial agonist. Ipsapirone (TVX Q 7821) also exhibits 5-HT1A receptor antagonistic effect, and only at high doses it can also produce an inhibitory effect on 5-HT2 and the α1-adrenergic function.	price>
R-R-3384	Iprindole CAS No.5560-72-5	Iprindole/CAS No.5560-72-5, a tricyclic indole antidepressant, is a weak inhibitor of the uptake of noradrenaline and 5-HT.	price>
R-R-3385	cis-(Z)-Flupentixol dihydrochloride CAS No.51529-01-2	cis-(Z)-Flupentixol dihydrochloride/CAS No.51529-01-2 is a potent and selective DA D1/D2 receptor antagonist, with Ki values of 0.38 nM and 7 nM for D2 receptor and 5-HT2A, respectively.	price>
R-C-1686	MK 0557 CAS:328232-95-7	MK-0557 is a highly selective,orally administered neuropeptide NPY5R antagonist,could limit weight regain after very-low-calorie diet(VLCD)-induced weight loss.Neuropeptide Y(NPY)is a potent orexigenic neuropeptide,and antagonism of NPY Y1 and NPY Y5 receptors(NPYxR)is considered a potentially important anti-obesity drug target.	price>
R-R-3386	Prucalopride-13C,d3 CAS No.2140306-00-7	Prucalopride-13C,d3/CAS No.2140306-00-7 is the 13C- and deuterium labeled Prucalopride.	price>
R-R-3387	LY 344864 racemate CAS No.186543-64-6	LY 344864 racemate/CAS No.186543-64-6 is a 5-HT1F receptor agonist extracted from patent US 5708187 A.	price>
R-R-3388	Hydroxy ziprasidone CAS No.884305-08-2	Hydroxy ziprasidone/CAS No.884305-08-2 is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a combined 5-HT (serotonin) and dopamine receptor antagonist.	price>
R-R-3389	Gepirone-d8 CAS No.2749331-28-8	Gepirone-d8/CAS No.2749331-28-8 is deuterium labeled Gepirone.	price>
R-R-3390	(Rac)-Rotigotine hydrochloride CAS No.102120-99-0	(Rac)-Rotigotine hydrochloride/CAS No.102120-99-0 is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial agonist of the 5-HT1A receptor, and an antagonist of the α2B-adrenergic receptor, with Kis of 0.71 nM, 4-15 nM, and 83 nM for the dopamine D3 receptor and D2, D5, D4 receptors, and dopamine D1 receptor.	price>
R-R-3391	Pardoprunox hydrochloride CAS No.269718-83-4	Pardoprunox (SLV-308) hydrochloride/CAS No.269718-83-4 is a partial dopamine D2 and D3 receptor partial agonist and a serotonin 5-HT1A receptor agonist, with pEC50s of 8, 9.2, and 6.3, respectively.	price>

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